SCHEMBL11116918

SCHEMBL11116918

CCOC(=O)C(Cc1ccc(C#N)cc1Cl)C(=O)OCC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
ALDH1A1 P00352 2/20 0.41
TSHR P16473 1/20 0.41
P2RX7 Q99572 1/20 0.41
GPR35 Q9HC97 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
PDCD1 Q15116 1/20 0.39
CD274 Q9NZQ7 1/20 0.39
PDK1 Q15118 1/20 0.39
PDK2 Q15119 1/20 0.39
PDK3 Q15120 1/20 0.39
PDK4 Q16654 1/20 0.39
AR P10275 2/20 0.38
FFAR1 O14842 1/20 0.38
MRGPRX4 Q96LA9 2/20 0.37
HTT P42858 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
TRPV4 Q9HBA0 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11114541 0.83 ALDH1A1 (0.48) ALDH1A1P2RX7PDK1PDK2PDK3
SCHEMBL533893 0.82 P2RX7 (0.41) ALDH1A1P2RX7GPR35PDK1PDK2
SCHEMBL9978726 0.81 CYP3A4 (0.61) CYP3A4CYP2C9ALDH1A1TSHRSMN1; SMN2
SCHEMBL16110186 0.81 PDCD1 (0.43) ALDH1A1P2RX7GPR35PDCD1CD274
SCHEMBL11116312 0.78 CYP4F2 (0.47) ALDH1A1P2RX7GPR35PDCD1CD274
SCHEMBL6119537 0.77 ALDH1A1 (0.41) ALDH1A1TSHRSMN1; SMN2PDCD1CD274
SCHEMBL2672524 0.77 MMP8 (0.50) ALDH1A1TSHRSMN1; SMN2NPSR1MAPT
SCHEMBL11450832 0.76 CYP3A4 (0.58) CYP3A4CYP2C9ALDH1A1TSHRSMN1; SMN2
SCHEMBL14107962 0.76 CYP2A6 (0.47) ALDH1A1TSHRP2RX7SMN1; SMN2PDK1
SCHEMBL2673394 0.75 ALDH1A1 (0.50) CYP3A4CYP2C9ALDH1A1TSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0038071-B1 NEW UNLABELLED AND RADIOACTIVE LABELLED DERIVATIVES OF BUTYLAMINO PROPIOPHENONE, THEIR PREPARATION, IMMUNOGENS OBTAINED FROM THE UNLABELLED DERIVATIVES AND A PROCESS FOR IMMUNOGEN PREPARATION, ANTISERA RAISED USING THE IMMUNOGENS AND A METHOD FOR RAISING ANTISERA, A RADIOIMMUNOASSAY METHOD AND A TEST KIT FOR USE IN THE ASSAY METHOD THE WELLCOME FOUNDATION LIMITED (GB) 1984-11-14 EP disclosed
US-4356165-A Bupropion radioimmunoassay, and kit BURROUGHS WELLCOME CO. (US) 1982-10-26 US disclosed
US-4355179-A Radioactive nuclide labeled propiophenone compounds BURROUGHS WELLCOME CO. (US) 1982-10-19 US disclosed
US-4347177-A Compounds and methods of making them BURROUGHS WELLCOME CO. (US) 1982-08-31 US disclosed
US-4347382-A 3H Labeled compounds BURROUGHS WELLCOME CO. (US) 1982-08-31 US disclosed
US-4347176-A Compounds and methods of making same BURROUGHS WELLCOME CO. (US) 1982-08-31 US disclosed
US-4347178-A Compounds and methods of making BURROUGHS WELLCOME CO. (US) 1982-08-31 US disclosed
EP-0038071-A2 New unlabelled and radioactive labelled derivatives of butylamino propiophenone, their preparation, immunogens obtained from the unlabelled derivatives and a process for immunogen preparation, antisera raised using the immunogens and a method for raising antisera, a radioimmunoassay method and a test kit for use in the assay method THE WELLCOME FOUNDATION LIMITED (GB) 1981-10-21 EP disclosed