SCHEMBL11116601

SCHEMBL11116601

CCOC(=O)C1(c2ccc(F)cc2C)CCN(S(=O)(=O)c2ccc(C)cc2)CC1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.48
CYP2C19 P33261 2/20 0.48
KMT2A Q03164 2/20 0.47
LMNA P02545 3/20 0.46
HTT P42858 1/20 0.46
OPRM1 P35372 2/20 0.46
USP2 O75604 1/20 0.45
TP53 P04637 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
HSD17B10 Q99714 1/20 0.45
PKM P14618 1/20 0.44
GAA P10253 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11133437 0.92 ALDH1A1 (0.48) ALDH1A1CYP2C19KMT2ALMNAHTT
SCHEMBL11127656 0.86 CYP2C19 (0.62) ALDH1A1CYP2C19KMT2ALMNAUSP2
SCHEMBL11113875 0.85 CYP2C19 (0.52) ALDH1A1CYP2C19KMT2ALMNAHTT
SCHEMBL11118092 0.80 CYP2C19 (0.55) ALDH1A1CYP2C19KMT2ALMNAHTT
SCHEMBL11392570 0.79 CYP2C19 (0.53) ALDH1A1CYP2C19KMT2ALMNAOPRM1
SCHEMBL11114152 0.78 ALDH1A1 (0.52) ALDH1A1CYP2C19KMT2ALMNAHTT
SCHEMBL6520496 0.78 ALDH1A1 (0.58) ALDH1A1CYP2C19KMT2ALMNAHTT
SCHEMBL11128806 0.78 CYP2C19 (0.62) ALDH1A1CYP2C19KMT2ALMNAUSP2
SCHEMBL11113941 0.77 SMN1; SMN2 (0.52) ALDH1A1KMT2ALMNAHTTGAA
SCHEMBL11119188 0.77 CYP2C19 (0.52) ALDH1A1CYP2C19KMT2ALMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0034415-B1 1-(CYCLOHEXYL OR CYCLOHEXENYL)-4-ARYL-4-PIPERIDINECARBOXYLIC ACID DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1984-05-30 EP disclosed
US-4369184-A ANTIHISTAMINES; HETEROCYCLIC NITRILES JANSSEN PHARMACEUTICA N.V. (BE) 1983-01-18 US disclosed
EP-0034415-A1 1-(Cyclohexyl or cyclohexenyl)-4-aryl-4-piperidinecarboxylic acid derivatives JANSSEN PHARMACEUTICA N.V. (BE) 1981-08-26 EP disclosed