SCHEMBL11118092

SCHEMBL11118092

CCOC(=O)C1(c2ccccc2OC)CCN(S(=O)(=O)c2ccc(C)cc2)CC1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.55
KMT2A Q03164 4/20 0.54
MEN1 O00255 3/20 0.54
GAA P10253 2/20 0.54
OXTR P30559 1/20 0.51
PKM P14618 1/20 0.51
APP P05067 3/20 0.50
PSEN1 P49768 1/20 0.49
PSEN2 P49810 1/20 0.49
APH1B Q8WW43 1/20 0.49
NCSTN Q92542 1/20 0.49
APH1A Q96BI3 1/20 0.49
PSENEN Q9NZ42 1/20 0.49
ALDH1A1 P00352 2/20 0.49
LMNA P02545 2/20 0.47
HTT P42858 1/20 0.47
MAPT P10636 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11114414 0.87 CYP2C19 (0.69) CYP2C19KMT2AMEN1GAAOXTR
SCHEMBL11113941 0.86 SMN1; SMN2 (0.52) KMT2AMEN1GAAAPPPSEN1
SCHEMBL11120207 0.86 CYP2C19 (0.58) CYP2C19KMT2AMEN1GAAOXTR
SCHEMBL11392570 0.84 CYP2C19 (0.53) CYP2C19KMT2AMEN1GAAOXTR
SCHEMBL11114152 0.83 ALDH1A1 (0.52) CYP2C19KMT2AMEN1GAAOXTR
SCHEMBL11116601 0.80 ALDH1A1 (0.48) CYP2C19KMT2AGAAPKMALDH1A1
SCHEMBL11133437 0.80 ALDH1A1 (0.48) CYP2C19KMT2AGAAPKMALDH1A1
SCHEMBL20790150 0.80 OPRM1 (0.50) KMT2AMEN1APPPSEN1PSEN2
SCHEMBL6520496 0.79 ALDH1A1 (0.58) CYP2C19KMT2AMEN1GAAPKM
SCHEMBL11118953 0.76 ADRA1D (0.53) CYP2C19KMT2AMEN1GAAOXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0034415-B1 1-(CYCLOHEXYL OR CYCLOHEXENYL)-4-ARYL-4-PIPERIDINECARBOXYLIC ACID DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1984-05-30 EP disclosed
US-4369184-A ANTIHISTAMINES; HETEROCYCLIC NITRILES JANSSEN PHARMACEUTICA N.V. (BE) 1983-01-18 US disclosed
EP-0034415-A1 1-(Cyclohexyl or cyclohexenyl)-4-aryl-4-piperidinecarboxylic acid derivatives JANSSEN PHARMACEUTICA N.V. (BE) 1981-08-26 EP disclosed