SCHEMBL11124692

SCHEMBL11124692

Cc1cccc(C(N)=CC#N)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.52
RECQL P46063 1/20 0.49
PDE4A P27815 3/20 0.41
PDE4B Q07343 3/20 0.41
PDE4C Q08493 3/20 0.41
PDE4D Q08499 3/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
GABRA1 P14867 1/20 0.39
GABRG2 P18507 1/20 0.39
GABRB3 P28472 1/20 0.39
GABRB2 P47870 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
ATM Q13315 1/20 0.38
ACHE P22303 1/20 0.38
HTR3E A5X5Y0 1/20 0.38
HTR3B O95264 1/20 0.38
HTR3A P46098 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11124682 1.00 PARP1 (0.52) PARP1RECQLPDE4APDE4BPDE4C
SCHEMBL21901287 1.00 PARP1 (0.52) PARP1RECQLPDE4APDE4BPDE4C
SCHEMBL17268849 0.80 GABRA1 (0.51) PARP1PDE4APDE4BPDE4CPDE4D
SCHEMBL11117845 0.79 PDE4A (0.65) PARP1RECQLPDE4APDE4BPDE4C
SCHEMBL11290195 0.79 PDE4A (0.65) PARP1RECQLPDE4APDE4BPDE4C
SCHEMBL11117847 0.79 PDE4A (0.65) PARP1RECQLPDE4APDE4BPDE4C
SCHEMBL11085889 0.79 RECQL (0.62) PARP1RECQLPDE4APDE4BPDE4C
SCHEMBL11083594 0.79 PARP1 (0.52) PARP1RECQLPDE4APDE4BPDE4C
SCHEMBL3958624 0.79 RECQL (0.49) RECQLPDE4APDE4BPDE4CPDE4D
SCHEMBL11072261 0.79 PARP1 (0.52) PARP1RECQLGABRA1GABRG2GABRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0129407-A2 Improvements in and relating to (3-aryl-5-isothiazolyl)ureas ELI LILLY AND COMPANY (US) 1984-12-27 EP disclosed