SCHEMBL11129792

SCHEMBL11129792

CC(C)(CCc1ccc(C(N)=O)cc1)NC[C@H](O)c1ccccc1F

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 13/20 0.45
ADRB1 P08588 13/20 0.45
DPP4 P27487 4/20 0.44
ADRB3 P13945 2/20 0.41
ADRA1D P25100 1/20 0.41
ADRA1A P35348 1/20 0.41
ADRA1B P35368 1/20 0.41
CASR P41180 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11122771 1.00 ADRB2 (0.45) ADRB2ADRB1DPP4ADRB3ADRA1D
Hydrochloric Acid SCHEMBL8855378 0.99 ADRB2 (0.44) ADRB2ADRB1DPP4ADRB3ADRA1D
SCHEMBL11136288 0.85 ADRB2 (0.53) ADRB2ADRB1CASR
SCHEMBL11136281 0.85 ADRB2 (0.53) ADRB2ADRB1CASR
Oxalic Acid SCHEMBL11451371 0.84 ADRB2 (0.43) ADRB2ADRB1CASR
SCHEMBL10770012 0.84 ADRB3 (0.48) ADRB2ADRB1DPP4ADRB3ADRA1D
Hydrochloric Acid SCHEMBL11134351 0.84 ADRB2 (0.54) ADRB2ADRB1CASR
SCHEMBL3366477 0.84 ADRB3 (0.48) ADRB2ADRB1DPP4ADRB3ADRA1D
Hydrochloric Acid SCHEMBL10766903 0.83 ADRB3 (0.49) ADRB2ADRB1DPP4ADRB3ADRA1D
Hydrochloric Acid SCHEMBL10766900 0.83 ADRB3 (0.49) ADRB2ADRB1DPP4ADRB3ADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0047536-B1 SUBSTITUTED PROPYLAMINES ELI LILLY AND COMPANY (US) 1984-06-27 EP disclosed
EP-0007206-B1 PHENETHANOLAMINES, THEIR FORMULATIONS, PREPARATION AND USE ELI LILLY AND COMPANY (US) 1983-02-23 EP disclosed
EP-0047536-A2 Substituted propylamines ELI LILLY AND COMPANY (US) 1982-03-17 EP disclosed
EP-0007206-A1 Phenethanolamines, their formulations, preparation and use ELI LILLY AND COMPANY (US) 1980-01-23 EP disclosed