SCHEMBL1114108

SCHEMBL1114108

NS(=O)(=O)C1=CC=CC(NC2CCNC2)([N+](=O)[O-])C1Sc1ccccc1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4215300 0.79
SCHEMBL1114260 0.75 CA12 (0.32)
SCHEMBL6533266 0.65 BCL2L1 (0.31)
SCHEMBL1114110 0.62 CA2 (0.36)
SCHEMBL1700282 0.58 MAPT (0.50)
SCHEMBL1700017 0.58 MAPT (0.50)
SCHEMBL1112453 0.58 KDM1A (0.47)
SCHEMBL1546166 0.56 HDAC4 (0.51)
Hydrochloric Acid SCHEMBL6582044 0.56 KMT2A (0.67)
SCHEMBL7899199 0.56 SLC18A3 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2279174-A2 ARYLSULFONAMIDE COMPOUNDS, COMPOSITIONS AND METHODS OF USE Genentech, Inc. (US) 2011-02-02 EP disclosed
WO-2009143246-A2 ARYLSULFONAMIDE COMPOUNDS, COMPOSITIONS AND METHODS OF USE GENENTECH, INC. (US) 2009-11-26 WO disclosed