SCHEMBL11144615

SCHEMBL11144615

COc1ccc(CC(C)Cn2ccnc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 8/20 0.60
ALDH1A1 P00352 2/20 0.56
CYP3A4 P08684 2/20 0.56
MAPT P10636 2/20 0.56
TDP1 Q9NUW8 2/20 0.56
MEN1 O00255 2/20 0.56
KMT2A Q03164 2/20 0.56
TP53 P04637 1/20 0.56
CYP1A2 P05177 1/20 0.56
TSHR P16473 1/20 0.56
MAPK1 P28482 1/20 0.56
HSD17B10 Q99714 1/20 0.56
CYP2C9 P11712 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
TRPM8 Q7Z2W7 1/20 0.56
ORAI1 Q96D31 1/20 0.55
CYP19A1 P11511 3/20 0.53
ATM Q13315 1/20 0.51
CYP11B1 P15538 1/20 0.51
IDO1 P14902 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11145829 0.85 CACNA1B (0.49) TBXAS1KMT2ACYP19A1CYP11B1
SCHEMBL11145004 0.84 CYP2A6 (0.52) TBXAS1CYP3A4TDP1MEN1KMT2A
SCHEMBL11149487 0.84 CYP19A1 (0.51) TBXAS1CYP19A1CYP11B1IDO1
SCHEMBL11158462 0.84 CYP19A1 (0.51) CYP3A4MAPK1CYP19A1CYP11B1IDO1
Hydrochloric Acid SCHEMBL11147406 0.84 CACNA1B (0.48) TBXAS1KMT2ACYP19A1CYP11B1
SCHEMBL11146917 0.83 ACACB (0.50) TBXAS1ALDH1A1MEN1KMT2AMAPK1
Hydrochloric Acid SCHEMBL11149860 0.83 CYP2A6 (0.51) TBXAS1CYP3A4TDP1MEN1KMT2A
SCHEMBL11285064 0.82 CYP19A1 (0.57) TBXAS1ALDH1A1CYP3A4MAPTTDP1
SCHEMBL10892777 0.82 TBXAS1 (0.79) TBXAS1
SCHEMBL11432172 0.82 QPCT (0.49) ALDH1A1CYP3A4MAPTTDP1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0009683-B1 BASIC PHENYL ETHERS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THE PREPARATION OF THESE ETHERS AND COMPOSITIONS MERCK PATENT GmbH (DE) 1983-08-10 EP disclosed
EP-0009683-A1 Basic phenyl ethers, pharmaceutical compositions containing them and the preparation of these ethers and compositions MERCK PATENT GmbH (DE) 1980-04-16 EP disclosed