SCHEMBL1114609

SCHEMBL1114609

Oc1c(Br)cc(C2=NCON2Cc2ccccc2C(F)(F)F)cc1Br

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.36
KDM4E B2RXH2 5/20 0.36
ATM Q13315 2/20 0.36
HTT P42858 2/20 0.36
TSHR P16473 2/20 0.36
KMT2A Q03164 3/20 0.35
MEN1 O00255 2/20 0.35
COMT P21964 1/20 0.35
TDP1 Q9NUW8 2/20 0.34
NPSR1 Q6W5P4 2/20 0.34
GAA P10253 1/20 0.34
ALOX15 P16050 2/20 0.34
MAPT P10636 1/20 0.34
POLB P06746 2/20 0.34
SIRT2 Q8IXJ6 1/20 0.34
SIRT1 Q96EB6 1/20 0.34
NR1H2 P55055 1/20 0.34
NR1H3 Q13133 1/20 0.34
PHGDH O43175 1/20 0.34
EPHX2 P34913 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1114336 0.87 KDM4E (0.39) ALDH1A1KDM4EATMHTTKMT2A
SCHEMBL1114610 0.67 ALDH1A1 (0.34) ALDH1A1KDM4EATMTSHRKMT2A
SCHEMBL30482351 0.64 KDM4E (0.38) ALDH1A1KDM4EATMHTTTSHR
SCHEMBL1114927 0.63 KMT2A (0.49) KDM4EKMT2AMEN1MAPTEPHX2
SCHEMBL30482302 0.62 KDM4E (0.36) ALDH1A1KDM4EATMKMT2AMEN1
SCHEMBL15055647 0.61 KMT2A (0.47) ALDH1A1KDM4EATMTSHRKMT2A
SCHEMBL20818003 0.58 MKNK1 (0.46) ALDH1A1KDM4EATMKMT2AMEN1
SCHEMBL20817931 0.58 TDP1 (0.44) ALDH1A1KDM4EATMKMT2ACOMT
SCHEMBL27858676 0.58 COMT (0.46) ALDH1A1KDM4EATMTSHRKMT2A
SCHEMBL31669175 0.57 ALDH1A1 (0.74) ALDH1A1KDM4EATMTSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2278879-A2 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING OXADIAZOLE DERIVATIVES Institute for OneWorld Health (US) 2011-02-02 EP claimed
WO-2009131957-A2 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING OXADIAZOLE DERIVATIVES INSTITUTE FOR ONEWORLD HEALTH (US) 2009-10-29 WO claimed