SCHEMBL1114336

SCHEMBL1114336

Oc1c(Cl)cc(C2=NCON2Cc2ccccc2C(F)(F)F)cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.39
ATM Q13315 3/20 0.39
ALDH1A1 P00352 3/20 0.39
NR1H2 P55055 3/20 0.38
NR1H3 Q13133 3/20 0.38
HSD17B13 Q7Z5P4 7/20 0.38
HTT P42858 1/20 0.36
P2RX7 Q99572 1/20 0.36
KMT2A Q03164 2/20 0.35
TDP1 Q9NUW8 3/20 0.35
NPSR1 Q6W5P4 2/20 0.35
MEN1 O00255 1/20 0.35
COMT P21964 1/20 0.35
RECQL P46063 1/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1114609 0.87 ALDH1A1 (0.36) KDM4EATMALDH1A1NR1H2NR1H3
SCHEMBL4372432 0.70 HSD17B13 (0.43) KDM4EATMALDH1A1NR1H2NR1H3
SCHEMBL1114553 0.69 MGLL (0.39) ALDH1A1
SCHEMBL1114833 0.67 HSD17B13 (0.38) KDM4EATMALDH1A1NR1H2NR1H3
SCHEMBL4355638 0.67 UTS2R (0.51) KDM4EATMALDH1A1HSD17B13P2RX7
SCHEMBL3980590 0.62 KDM4E (0.53) KDM4EATMALDH1A1NR1H2NR1H3
SCHEMBL15055647 0.61 KMT2A (0.47) KDM4EATMALDH1A1KMT2ATDP1
SCHEMBL4359436 0.61 GAA (0.44) KDM4EALDH1A1HSD17B13HTTP2RX7
SCHEMBL28221686 0.58 ALDH1A1 (0.48) KDM4EATMALDH1A1NR1H2NR1H3
SCHEMBL1491106 0.58 KDM4E (0.46) KDM4EATMALDH1A1NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2278879-A2 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING OXADIAZOLE DERIVATIVES Institute for OneWorld Health (US) 2011-02-02 EP claimed
WO-2009131957-A2 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING OXADIAZOLE DERIVATIVES INSTITUTE FOR ONEWORLD HEALTH (US) 2009-10-29 WO claimed
EP-2278879-A2 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING OXADIAZOLE DERIVATIVES Institute for OneWorld Health (US) 2011-02-02 EP disclosed
WO-2009131957-A2 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING OXADIAZOLE DERIVATIVES INSTITUTE FOR ONEWORLD HEALTH (US) 2009-10-29 WO disclosed