SCHEMBL111493

SCHEMBL111493

CC(=O)C(N)(CSSCC(N)C(=O)O)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 6/20 0.41
NOS1 P29475 4/20 0.41
NOS3 P29474 3/20 0.41
KIF11 P52732 9/20 0.36
ARG1 P05089 1/20 0.34
ARG2 P78540 1/20 0.34
DNMT1 P26358 1/20 0.34
GRIK1 P39086 1/20 0.33
MEN1 O00255 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33
SLC7A5 Q01650 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20816349 1.00 NOS2 (0.41) NOS2NOS1NOS3KIF11ARG1
SCHEMBL6130506 0.87 NOS2 (0.39) NOS2NOS1NOS3KIF11ARG1
SCHEMBL20456896 0.84 NOS2 (0.37) NOS2NOS1NOS3KIF11ARG1
SCHEMBL9326098 0.84 KIF11 (0.36) NOS2NOS1NOS3KIF11ARG1
SCHEMBL10422578 0.84 KIF11 (0.36) NOS2NOS1NOS3KIF11ARG1
SCHEMBL121974 0.84 SMN1; SMN2 (0.34) NOS2NOS1NOS3MEN1KMT2A
SCHEMBL3921490 0.84 SMN1; SMN2 (0.34) NOS2NOS1NOS3MEN1KMT2A
SCHEMBL15757119 0.82 KIF11 (0.33) NOS2NOS1NOS3KIF11ARG1
SCHEMBL7115160 0.82 KIF11 (0.33) NOS2NOS1NOS3KIF11ARG1
SCHEMBL9810276 0.82 KIF11 (0.33) NOS2NOS1NOS3KIF11ARG1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 583 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4003906-A1 PEPTIDE-LOADED CARRIER SYSTEMS AND USES THEREOF Academia Sinica (TW) 2022-06-01 EP claimed
WO-2021021861-A1 PEPTIDE-LOADED CARRIER SYSTEMS AND USES THEREOF ACADEMIA SINICA (TW) 2021-02-04 WO claimed
WO-2020150499-A1 METHODS TO TAG AND ISOLATE CELLS INFECTED WITH THE HUMAN IMMUNODEFICIENCY VIRUS FRED HUTCHINSON CANCER RESEARCH CENTER (US) 2020-07-23 WO claimed
WO-2019027834-A1 COMPOSITIONS AND METHOD FOR ESTABLISHING ORGANOID CULTURES FROM CRYOGENICALLY PRESERVED TISSUE THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2019-02-07 WO claimed
EP-3071027-A1 ASSAY-READY FROZEN CELL AND METHOD FOR MINIMIZING VARIABILITY IN THE PERFORMANCE THEREOF Centre National de la Recherche Scientifique (C.N.R.S.) (FR) 2016-09-28 EP claimed
WO-2015077523-A1 ASSAY-READY FROZEN CELL AND METHOD FOR MINIMIZING VARIABILITY IN THE PERFORMANCE THEREOF LE CENTRE NATIONALE DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2015-05-28 WO claimed
US-5415870-A Layers of acid, alkali carbonate and alkali metal salt of acid Gergely, Gerhard (AT) 1995-05-16 US claimed
JP-58092622-A None JP disclosed
EP-4303228-B1 LONG-ACTING COAGULATION FACTOR VII AND METHODS OF PRODUCING SAME OPKO BIOLOGICS LTD (IL) 2026-05-27 EP disclosed
US-12516130-B2 Single-domain antibody for targeting prostate specific membrane antigen (PSMA) NATIONAL INSTITUTE OF BIOTECHNOLOGY IN THE NEGEV LTD. (IL) 2026-01-06 US disclosed
US-12459982-B2 Methods of producing long acting CTP-modified growth hormone polypeptides OPKO BIOLOGISTICS LTD. (IL) 2025-11-04 US disclosed
EP-3681511-B1 COMPOSITION AND METHOD FOR A PREBIOTIC DELIVERY SYSTEM TARGETED TO PROBIOTIC BACTERIA TECHNION RES & DEV FOUNDATION (IL) 2025-10-29 EP disclosed
US-12391944-B2 Magnetic inorganic iron-based nanoparticles BAR-ILAN UNIVERSITY (IL) 2025-08-19 US disclosed
WO-1998023611-A1 2-IMIDAZOLINYLAMINOBENZOXAZOLE COMPOUNDS USEFUL AS ALPHA-2 ADRENOCEPTOR AGONISTS THE PROCTER & GAMBLE COMPANY (US) 1998-06-04 WO disclosed
WO-1998023610-A1 2-IMIDAZOLINYLAMINOINDOLE COMPOUNDS USEFUL AS ALPHA-2 ADRENOCEPTOR AGONISTS THE PROCTER & GAMBLE COMPANY (US) 1998-06-04 WO disclosed
WO-1998023612-A1 2-IMIDAZOLINYLAMINOBENZOTHIAZOLE COMPOUNDS USEFUL AS ALPHA-2 ADRENOCEPTOR AGONISTS THE PROCTER & GAMBLE COMPANY (US) 1998-06-04 WO disclosed
WO-1998023596-A1 GUANIDINYL HETEROCYCLE COMPOUNDS USEFUL AS ALPHA-2 ADRENOCEPTOR AGONISTS THE PROCTER & GAMBLE COMPANY (US) 1998-06-04 WO disclosed
WO-1998023591-A1 GUANIDINYLAMINO HETEROCYCLE COMPOUNDS USEFUL AS ALPHA-2 ADRENOCEPTOR AGONISTS THE PROCTER & GAMBLE COMPANY (US) 1998-06-04 WO disclosed
WO-1998023609-A1 2-IMIDAZOLINYLAMINOINDAZOLE COMPOUNDS USEFUL AS ALPHA-2 ADRENOCEPTOR AGONISTS THE PROCTER & GAMBLE COMPANY (US) 1998-06-04 WO disclosed
JP-S5892622-A PHARMACEUTICAL PREPARATION CONTAINING STABLY COMPOUNDED INTERFERON SUNSTAR INC 1983-06-02 JP disclosed