SCHEMBL11149709

SCHEMBL11149709

CC(Br)CCN1C(=O)C(=O)c2ccccc21

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 7/20 0.67
BCHE P06276 2/20 0.67
ALDH1A1 P00352 7/20 0.59
ALDH3A1 P30838 5/20 0.59
ALDH2 P05091 4/20 0.59
CDC25A P30304 1/20 0.57
TGM2 P21980 1/20 0.57
PARK7 Q99497 1/20 0.56
PKM P14618 1/20 0.54
TP53 P04637 1/20 0.52
AGTR1 P30556 1/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
CHRM1 P11229 2/20 0.51
CA1 P00915 1/20 0.51
CA2 P00918 1/20 0.51
CHRM5 P08912 1/20 0.50
CHRM3 P20309 1/20 0.50
TTR P02766 1/20 0.50
MAOA P21397 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL281962 0.91 ALDH1A1 (0.64) CES1BCHEALDH1A1ALDH3A1ALDH2
SCHEMBL578329 0.87 CES1 (0.71) CES1BCHEALDH1A1ALDH3A1ALDH2
SCHEMBL5428316 0.83 CES1 (0.65) CES1BCHEALDH1A1ALDH3A1ALDH2
SCHEMBL4309242 0.82 ALDH1A1 (0.59) ALDH1A1MAOB
SCHEMBL19924204 0.81 CES1 (1.00) CES1BCHEALDH1A1ALDH3A1ALDH2
SCHEMBL3016508 0.78 CES1 (0.79) CES1BCHEALDH1A1ALDH3A1ALDH2
SCHEMBL10685462 0.78 CES1 (1.00) CES1BCHEALDH1A1ALDH3A1ALDH2
SCHEMBL10682318 0.78 CES1 (0.67) CES1BCHEALDH1A1ALDH3A1ALDH2
SCHEMBL25119569 0.78 CES1 (0.85) CES1BCHEALDH1A1ALDH3A1ALDH2
SCHEMBL10681723 0.77 CES1 (0.65) CES1BCHEALDH1A1ALDH3A1ALDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4382934-A ANTIALLERGENS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1983-05-10 US disclosed
EP-0010398-B1 ISATIN DERIVATIVES, PROCESSES FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1983-04-27 EP disclosed
EP-0010398-A1 Isatin derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1980-04-30 EP disclosed