SCHEMBL11152007

SCHEMBL11152007

CCOC(=O)C=Cc1ccc(NCCCCC2CCCCCC2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA7 P43166 1/20 0.48
CA9 Q16790 1/20 0.48
CA14 Q9ULX7 1/20 0.48
CYP3A4 P08684 1/20 0.44
TTR P02766 1/20 0.43
DPP4 P27487 1/20 0.43
RAB9A P51151 1/20 0.42
CNR1 P21554 1/20 0.42
CNR2 P34972 1/20 0.42
EPHX2 P34913 1/20 0.41
ESR1 P03372 1/20 0.41
METAP2 P50579 1/20 0.40
HDAC1 Q13547 2/20 0.40
KCNH2 Q12809 1/20 0.40
MAOB P27338 1/20 0.40
LMNA P02545 2/20 0.39
BCHE P06276 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11152011 1.00 CA12 (0.48) CA12CA1CA2CA7CA9
SCHEMBL846845 0.85 CA12 (0.53) CA12CA1CA2CA7CA9
SCHEMBL11156911 0.85 CA12 (0.53) CA12CA1CA2CA7CA9
SCHEMBL11186707 0.83 RAB9A (0.40) CYP3A4RAB9ACNR1KCNH2LMNA
SCHEMBL11186705 0.83 RAB9A (0.40) CYP3A4RAB9ACNR1KCNH2LMNA
SCHEMBL11229892 0.81 CA12 (0.57) CA12CA1CA2CA7CA9
SCHEMBL11229891 0.81 CA12 (0.57) CA12CA1CA2CA7CA9
SCHEMBL11262554 0.81 CA12 (0.57) CA12CA1CA2CA7CA9
SCHEMBL11262552 0.81 CA12 (0.57) CA12CA1CA2CA7CA9
SCHEMBL11147830 0.80 MAPT (0.48) RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4388459-A HYPOLIPIDEMIC, ANTIATHEROSCLEROTIC AMERICAN CYANAMID COMPANY (US) 1983-06-14 US disclosed
US-4259352-A 4-[Cycloalkyl- or cycloalkenyl-amino(cycloalkyl- or cycloalkenyl-alkenyl)amino]phenyl compounds, useful as hypolipidemic and antiatherosclerotic agents AMERICAN CYANAMID COMPANY (US) 1981-03-31 US disclosed
EP-0003663-A2 Amino-substituted phenyl and heteroaryl compounds, process for their preparation and pharmaceutical compositions containing them AMERICAN CYANAMID COMPANY (US) 1979-08-22 EP disclosed