SCHEMBL11178024

SCHEMBL11178024

COc1ccc(-c2nc(C(O)(C(F)(F)F)C(F)(F)F)n(C)c2-c2ccc(OC)cc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 2/20 0.44
LMNA P02545 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
PTGS2 P35354 1/20 0.38
MEN1 O00255 4/20 0.38
KMT2A Q03164 4/20 0.38
MAPT P10636 2/20 0.37
GAA P10253 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
SCN5A Q14524 1/20 0.36
MAPK13 O15264 1/20 0.36
MAPK12 P53778 1/20 0.36
MAPK11 Q15759 1/20 0.36
MAPK14 Q16539 1/20 0.36
GRIA1 P42261 1/20 0.36
CACNG2 Q9Y698 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9263043 0.84 ALDH1A1 (0.43) MLYCDLMNANPSR1KDM4EALDH1A1
SCHEMBL11176149 0.75 CNR1 (0.46) PTGS2MAPK13MAPK12MAPK11MAPK14
SCHEMBL11164503 0.75 ALDH1A1 (0.39) LMNANPSR1KDM4EALDH1A1TDP1
SCHEMBL10989518 0.72 ALDH1A1 (0.47) LMNANPSR1KDM4EALDH1A1TDP1
SCHEMBL5443200 0.72 ALDH1A1 (0.47) LMNANPSR1KDM4EALDH1A1TDP1
SCHEMBL7085313 0.70 MAPK14 (0.59) LMNANPSR1KDM4EALDH1A1TDP1
SCHEMBL27881874 0.69 LMNA (0.59) LMNANPSR1KDM4EALDH1A1TDP1
SCHEMBL11169683 0.69 KMT2A (0.44) LMNANPSR1KDM4EALDH1A1TDP1
SCHEMBL11165161 0.69 NOX1 (0.53) MLYCDLMNANPSR1KDM4EALDH1A1
SCHEMBL21852751 0.68 ALDH1A1 (0.67) LMNANPSR1KDM4EALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4372964-A ANAGESIC, ANTIARTHRITIC E. I. DU PONT DE NEMOURS AND COMPANY (US) 1983-02-08 US disclosed
EP-0032113-A2 Antiinflammatory 4,5-diaryl-alpha-(polyhaloalkyl)-1H-imidazole-2-methanols E.I. DU PONT DE NEMOURS AND COMPANY (US) 1981-07-15 EP disclosed