SCHEMBL11180959

SCHEMBL11180959

CC(c1cccc(O)c1)N1CCCC1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.52
CYP2D6 P10635 3/20 0.50
MBTD1 Q05BQ5 1/20 0.49
L3MBTL3 Q96JM7 1/20 0.49
ADRB1 P08588 2/20 0.47
ADRA1A P35348 2/20 0.47
MIF P14174 1/20 0.47
HTR2A P28223 1/20 0.47
HTR2B P41595 1/20 0.47
MC4R P32245 1/20 0.44
OPRM1 P35372 2/20 0.41
OPRD1 P41143 1/20 0.41
OPRK1 P41145 1/20 0.41
OPRL1 P41146 1/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C9 P11712 2/20 0.41
KCNA5 P22460 2/20 0.41
CYP2C19 P33261 2/20 0.41
KCNH2 Q12809 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11191579 0.98 ACHE (0.55) ACHECYP2D6MBTD1L3MBTL3ADRB1
SCHEMBL11189977 0.98 ACHE (0.55) ACHECYP2D6MBTD1L3MBTL3ADRB1
SCHEMBL14701580 0.81 CYP2D6 (0.53) ACHECYP2D6MBTD1L3MBTL3MC4R
SCHEMBL26575270 0.79 CYP2D6 (0.50) ACHECYP2D6MBTD1L3MBTL3MC4R
SCHEMBL31669513 0.79 CHRNA1 (0.51) ACHECYP2D6MBTD1L3MBTL3MC4R
SCHEMBL17319361 0.79 SLC6A2 (0.53) ACHECYP2D6MBTD1L3MBTL3MC4R
SCHEMBL15332985 0.78 ACHE (0.49) ACHECYP2D6MBTD1L3MBTL3MC4R
SCHEMBL11172155 0.78 OPRM1 (0.46) CYP2D6ADRB1ADRA1AOPRM1OPRD1
SCHEMBL30341013 0.77 SLC6A2 (0.54) ACHECYP2D6MBTD1L3MBTL3MC4R
SCHEMBL8983562 0.77 CYP2D6 (0.83) CYP2D6MC4ROPRM1OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107417574-A 2,4 disubstituted benzene ethanone compounds and its optical isomer, pharmaceutically acceptable salt and application 浙江省医学科学院 2017-12-01 CN disclosed
EP-0024510-B1 PHENOXYPROPYL AMINE DERIVATIVES, PROCESS FOR THEIR PREPARATION, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM TEIKOKU HORMONE MFG. CO., LTD. (JP) 1983-10-19 EP disclosed
US-4293557-A AMIDES TEIKOKU HORMONE MFG. CO., LTD. (JP) 1981-10-06 US disclosed
EP-0024510-A1 Phenoxypropyl amine derivatives, process for their preparation, and pharmaceutical compositions containing them TEIKOKU HORMONE MFG. CO., LTD. (JP) 1981-03-11 EP disclosed