SCHEMBL1119908

SCHEMBL1119908

COc1cccc(CN(C)C(CO)c2ccc3ccccc3c2)c1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.49
CALM1 P0DP23 1/20 0.44
CAMKK2 Q96RR4 1/20 0.44
ABCB11 O95342 1/20 0.44
ALDH1A1 P00352 4/20 0.43
MEN1 O00255 3/20 0.43
KDM4E B2RXH2 3/20 0.43
LMNA P02545 2/20 0.43
MTNR1A P48039 1/20 0.43
MTNR1B P49286 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
TDP1 Q9NUW8 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
UTS2R Q9UKP6 1/20 0.41
AOC3 Q16853 2/20 0.40
HSD17B2 P37059 1/20 0.40
GAA P10253 1/20 0.40
TAAR1 Q96RJ0 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL747464 0.84 KMT2A (0.42) KMT2ACALM1CAMKK2ALDH1A1MEN1
SCHEMBL1119877 0.84 AOC3 (0.40) UTS2RAOC3TAAR1
SCHEMBL4740860 0.78 ABCB11 (0.47) KMT2AABCB11MEN1
SCHEMBL12633238 0.78 KMT2A (0.55) KMT2ACALM1CAMKK2ALDH1A1MEN1
SCHEMBL1119907 0.78 KMT2A (0.55) KMT2ACALM1CAMKK2ALDH1A1MEN1
SCHEMBL13566617 0.77 KMT2A (0.53) KMT2ACALM1CAMKK2ABCB11ALDH1A1
SCHEMBL27812151 0.75 KMT2A (0.52) KMT2AALDH1A1MEN1KDM4EMTNR1A
SCHEMBL5571032 0.74 SLC6A2 (0.47) KMT2AAOC3
SCHEMBL27812152 0.73 KMT2A (0.49) KMT2ACALM1CAMKK2ALDH1A1MEN1
SCHEMBL1956804 0.72 IDO1 (0.48) KMT2AMTNR1AMTNR1BSMN1; SMN2TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2280956-A2 PROCESSES FOR PREPARING TETRAHYDROISOQUINOLINES Bristol-Myers Squibb Company (US) 2011-02-09 EP disclosed
WO-2009149259-A2 PROCESSES FOR PREPARING TETRAHYDROISOQUINOLINES BRISTOL-MYERS SQUIBB COMPANY (US) 2009-12-10 WO disclosed