SCHEMBL4740860

SCHEMBL4740860

COc1ccc2cc(C(CCO)N(C)Cc3ccccc3)ccc2c1

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 1/20 0.47
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
CLK1 P49759 1/20 0.44
DYRK1A Q13627 1/20 0.44
AKR1C3 P42330 6/20 0.43
AKR1C2 P52895 6/20 0.43
PTGS1 P23219 3/20 0.43
AKR1C1 Q04828 1/20 0.43
PTGS2 P35354 3/20 0.43
CDC42 P60953 1/20 0.43
RAC1 P63000 1/20 0.43
CYP1A2 P05177 1/20 0.43
TSHR P16473 1/20 0.43
SLC22A6 Q4U2R8 1/20 0.43
ACHE P22303 2/20 0.41
NPC1 O15118 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4740861 0.82 TNF (0.50) MEN1KMT2AACHENPC1
SCHEMBL5164752 0.78 HTR2A (0.47) MEN1KMT2ATSHRNPC1POLB
SCHEMBL1119908 0.78 KMT2A (0.49) ABCB11MEN1KMT2A
SCHEMBL4739767 0.75 UTS2R (0.42) RXFP1CYP1A2TSHRPOLB
SCHEMBL3978356 0.73 UGT2B7 (0.43) MEN1KMT2ACYP1A2TSHRACHE
SCHEMBL17073799 0.72 TSHR (0.51) ABCB11MEN1KMT2AAKR1C3AKR1C2
SCHEMBL8075567 0.71 ABCB11 (0.48) ABCB11MEN1KMT2AAKR1C3AKR1C2
SCHEMBL6091855 0.71 AOC3 (0.50) MEN1KMT2ACYP1A2TSHR
SCHEMBL13986008 0.70 SLC6A2 (0.53) MEN1KMT2ATSHRACHENPC1
SCHEMBL9050772 0.70 ABCB11 (0.59) ABCB11AKR1C3AKR1C2PTGS1AKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008081477-A1 3-ARYLOXY 3-SUBSTITUTED PROPANAMINES NATCO PHARMA LIMITED (IN) 2008-07-10 WO disclosed