SCHEMBL11201072

SCHEMBL11201072

c1ccc(CN2Cc3ccccc3C2)c(CN2CCOCC2)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A13 Q16696 7/20 0.62
ALDH1A1 P00352 3/20 0.53
CYP2C9 P11712 2/20 0.53
KMT2A Q03164 2/20 0.53
ALOX15 P16050 1/20 0.53
HSD17B10 Q99714 1/20 0.53
MEN1 O00255 1/20 0.53
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C19 P33261 1/20 0.50
KDM4E B2RXH2 2/20 0.49
ADRA2A P08913 1/20 0.49
ADRA2B P18089 1/20 0.49
ADRA2C P18825 1/20 0.49
TMEM97 Q5BJF2 1/20 0.49
SIGMAR1 Q99720 1/20 0.49
LMNA P02545 1/20 0.49
GAA P10253 1/20 0.49
MAPT P10636 1/20 0.49
TDP1 Q9NUW8 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11193326 0.89 CYP2A13 (0.75) CYP2A13ALDH1A1CYP2C9KMT2AALOX15
SCHEMBL11199250 0.81 ALDH1A1 (0.59) ALDH1A1KMT2AMEN1KDM4ELMNA
SCHEMBL4327006 0.80 MPO (0.75) CYP2A13ALDH1A1CYP2C9KMT2AALOX15
SCHEMBL4108619 0.80 CYP2A13 (0.69) CYP2A13ALDH1A1CYP2C9KMT2AALOX15
SCHEMBL111727 0.80 CYP2A13 (0.64) CYP2A13ALDH1A1CYP2C9KMT2AALOX15
SCHEMBL2251851 0.80 CYP2A13 (0.64) CYP2A13ALDH1A1CYP2C9KMT2AALOX15
SCHEMBL22711364 0.80 CYP2A13 (0.64) CYP2A13ALDH1A1CYP2C9KMT2AALOX15
SCHEMBL3738488 0.80 CYP2A13 (0.69) CYP2A13ALDH1A1CYP2C9KMT2AALOX15
SCHEMBL3730392 0.79 CYP2A13 (0.67) CYP2A13ALDH1A1CYP2C9KMT2AALOX15
SCHEMBL10787841 0.79 MPO (0.72) CYP2A13ALDH1A1CYP2C9KMT2AALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4333932-A DIHYDROISOINDOLES, HYPOGLYCEMIC, ANTIDIABETIC PFIZER INC. (US) 1982-06-08 US claimed
EP-0010896-A1 Organic diamine compounds for use as oral hypoglycemic agents and pharmaceutical compositions thereof PFIZER INC. (US) 1980-05-14 EP claimed
US-4414220-A HUPOGLYCEMIC, ANTIDIABETIC PFIZER INC. (US) 1983-11-08 US disclosed
US-4414220-A HUPOGLYCEMIC, ANTIDIABETIC PFIZER INC. (US) 1983-11-08 US disclosed
US-4333932-A DIHYDROISOINDOLES, HYPOGLYCEMIC, ANTIDIABETIC PFIZER INC. (US) 1982-06-08 US disclosed
US-4333932-A DIHYDROISOINDOLES, HYPOGLYCEMIC, ANTIDIABETIC PFIZER INC. (US) 1982-06-08 US disclosed
US-4220650-A HYPOGLYCEMIC PFIZER INC. (US) 1980-09-02 US disclosed
US-4220650-A HYPOGLYCEMIC PFIZER INC. (US) 1980-09-02 US disclosed
EP-0010896-A1 Organic diamine compounds for use as oral hypoglycemic agents and pharmaceutical compositions thereof PFIZER INC. (US) 1980-05-14 EP disclosed