SCHEMBL11201229

SCHEMBL11201229

CC(=O)N1CCN(c2nc(N)c3c(C(C)C)csc3n2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 1/20 0.40
GBA1 P04062 1/20 0.39
HCRTR1 O43613 2/20 0.39
HCRTR2 O43614 2/20 0.39
PIK3CA P42336 3/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CASP6 P55212 1/20 0.37
GFER P55789 1/20 0.37
MAP4K4 O95819 1/20 0.37
HSP90AA1 P07900 1/20 0.37
ADRA1A P35348 2/20 0.36
ADRA1B P35368 2/20 0.36
ITGB2 P05107 1/20 0.36
ICAM1 P05362 1/20 0.36
ITGAL P20701 1/20 0.36
PIK3CD O00329 1/20 0.36
PIK3R1 P27986 1/20 0.36
PIK3CB P42338 1/20 0.36
PIK3CG P48736 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11202244 0.86 MAPT (0.47) PTPN11SMN1; SMN2NPSR1MEN1KMT2A
SCHEMBL11133041 0.84 HCRTR1 (0.51) PTPN11GBA1HCRTR1HCRTR2PIK3CA
SCHEMBL11206583 0.82 PTPN11 (0.41) PTPN11GBA1HCRTR1HCRTR2PIK3CA
SCHEMBL11201993 0.82 HCRTR1 (0.37) HCRTR1HCRTR2ITGB2ICAM1ITGAL
SCHEMBL11204218 0.81 KDM4E (0.41) HCRTR1HCRTR2SMN1; SMN2
Hydrochloric Acid SCHEMBL11198496 0.80 KDM4E (0.40) HCRTR1HCRTR2SMN1; SMN2
SCHEMBL11205242 0.71 MAPT (0.45) PTPN11SMN1; SMN2NPSR1MEN1KMT2A
SCHEMBL11206086 0.70 HCRTR1 (0.51) PTPN11GBA1HCRTR1HCRTR2PIK3CA
SCHEMBL11202336 0.70 MAPK1 (0.51) NPSR1MEN1KMT2A
SCHEMBL11202238 0.70 GBA1 (0.39) PTPN11GBA1PIK3CASMN1; SMN2CASP6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0082023-A2 Thienopyrimidine derivatives, their preparation and their medical use SANKYO COMPANY LIMITED (JP) 1983-06-22 EP disclosed