SCHEMBL11201993

SCHEMBL11201993

CC(C)c1csc2nc(N3CCN(C=O)CC3)nc(N)c12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.37
HCRTR2 O43614 2/20 0.37
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
MAPT P10636 1/20 0.36
MAPK1 P28482 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ELANE P08246 2/20 0.34
HRH4 Q9H3N8 2/20 0.33
HTR3A P46098 1/20 0.33
ADORA2A P29274 1/20 0.32
ITGB2 P05107 1/20 0.32
ICAM1 P05362 1/20 0.32
ITGAL P20701 1/20 0.32
KMT2A Q03164 1/20 0.31
HTR1A P08908 3/20 0.31
HTR2A P28223 3/20 0.31
HTR7 P34969 3/20 0.31
HTR6 P50406 3/20 0.31
DRD2 P14416 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11197939 0.84 HCRTR1 (0.49) HCRTR1HCRTR2KDM4EALDH1A1MAPT
SCHEMBL11201229 0.82 PTPN11 (0.40) HCRTR1HCRTR2ITGB2ICAM1ITGAL
SCHEMBL11202902 0.82 HCRTR1 (0.38) HCRTR1HCRTR2KDM4EALDH1A1MAPT
SCHEMBL11204218 0.81 KDM4E (0.41) HCRTR1HCRTR2KDM4EALDH1A1MAPT
SCHEMBL11202884 0.81 HCRTR1 (0.47) HCRTR1HCRTR2KDM4EALDH1A1MAPT
Hydrochloric Acid SCHEMBL11198496 0.81 KDM4E (0.40) HCRTR1HCRTR2KDM4EALDH1A1MAPT
SCHEMBL11201413 0.79 HCRTR1 (0.36) HCRTR1HCRTR2KDM4EALDH1A1MAPT
SCHEMBL11201137 0.79 ESR1 (0.39) KDM4EALDH1A1MAPTMAPK1L3MBTL1
SCHEMBL11203490 0.79 ELANE (0.36) KDM4EALDH1A1MAPTMAPK1L3MBTL1
SCHEMBL11202244 0.78 MAPT (0.47) KDM4EALDH1A1MAPTMAPK1ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0082023-A2 Thienopyrimidine derivatives, their preparation and their medical use SANKYO COMPANY LIMITED (JP) 1983-06-22 EP disclosed