SCHEMBL11201723

SCHEMBL11201723

CCc1sc2nc(N3CCNCC3)nc(NC)c2c1C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KHK P50053 3/20 0.39
HTR2A P28223 1/20 0.38
HRH1 P35367 1/20 0.37
USP2 O75604 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
HRH4 Q9H3N8 1/20 0.36
HTR2C P28335 2/20 0.35
ROCK2 O75116 1/20 0.35
PLK4 O00444 1/20 0.34
PAK4 O96013 1/20 0.34
CASP1 P29466 1/20 0.33
CASP4 P49662 1/20 0.33
CASP5 P51878 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
PDE5A O76074 1/20 0.33
P2RY12 Q9H244 1/20 0.33
GUSB P08236 1/20 0.33
ADRB1 P08588 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11203991 0.89 HTR2A (0.38) KHKHTR2AHRH1USP2SMN1; SMN2
SCHEMBL11205170 0.86 ALDH1A1 (0.42) KHKHRH1USP2SMN1; SMN2TDP1
SCHEMBL11203366 0.85 KHK (0.41) KHKHTR2AHRH1USP2SMN1; SMN2
SCHEMBL11202792 0.84 KHK (0.38) KHKHTR2AHRH1USP2SMN1; SMN2
SCHEMBL11202267 0.83 KDM4E (0.39) HTR2AHRH1USP2SMN1; SMN2TDP1
SCHEMBL11201110 0.83 HRH4 (0.36) HRH4KDM4EALDH1A1
SCHEMBL11197095 0.81 CETP (0.39) KHKHTR2AHRH1USP2SMN1; SMN2
SCHEMBL11200202 0.81 KHK (0.38) KHKHTR2AHRH1USP2SMN1; SMN2
SCHEMBL11201393 0.79 HRH1 (0.41) HRH1USP2SMN1; SMN2TDP1HRH4
SCHEMBL11197339 0.78 HTR2C (0.39) KHKHTR2AHRH1USP2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0082023-A2 Thienopyrimidine derivatives, their preparation and their medical use SANKYO COMPANY LIMITED (JP) 1983-06-22 EP disclosed