SCHEMBL11202198

SCHEMBL11202198

O=C(c1ccoc1)c1ccc2n1CCCC2C(=O)O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC42 P60953 3/20 0.59
RAC1 P63000 3/20 0.59
PTGS2 P35354 3/20 0.59
PTGS1 P23219 2/20 0.59
NPC1 O15118 1/20 0.59
CHRM3 P20309 1/20 0.59
OPRM1 P35372 1/20 0.59
RAB9A P51151 1/20 0.59
PAK1 Q13153 1/20 0.59
ABCC4 O15439 1/20 0.49
HTT P42858 1/20 0.49
BLM P54132 1/20 0.49
LMNA P02545 1/20 0.49
CYP1A2 P05177 1/20 0.49
NFKB1 P19838 1/20 0.49
MAPK1 P28482 1/20 0.49
CA4 P22748 5/20 0.38
CA9 Q16790 4/20 0.38
CA12 O43570 3/20 0.38
CA1 P00915 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11197022 0.96 PTGS2 (0.57) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL11661178 0.92 PTGS2 (0.69) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL11201371 0.83 PTGS2 (0.40) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL11195095 0.83 CDC42 (0.50) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL11194395 0.83 PTGS2 (0.84) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL11661267 0.80 PTGS2 (0.52) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL11206915 0.80 PTGS2 (0.40) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL11194207 0.80 NPC1 (0.65) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL11201477 0.80 CDC42 (0.65) CDC42RAC1PTGS2PTGS1NPC1
SCHEMBL11194044 0.80 PTGS2 (0.65) CDC42RAC1PTGS2PTGS1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4410534-A 3-Substituted-5,6,7,8-tetrahydropyrrolo[1,2-a]-pyridine-and 6,7,8,9-tetrahydro-5H-pyrrolo[1,2-a]-azepine carboxylic acid derivatives useful as blood platelet aggregation inhibitors SYNTEX (U.S.A.) INC. (US) 1983-10-18 US disclosed