SCHEMBL11206227

SCHEMBL11206227

O=C1C[C@H]2CCCC[C@@H]2CN1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.38
MAP3K14 Q99558 1/20 0.34
PDE4A P27815 6/20 0.33
PDE4B Q07343 6/20 0.33
PDE4C Q08493 6/20 0.33
PDE4D Q08499 6/20 0.33
CYP3A4 P08684 2/20 0.33
ALDH1A1 P00352 2/20 0.33
VEGFA P15692 1/20 0.33
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
ALOX15 P16050 1/20 0.33
CREBBP Q92793 1/20 0.33
KDM4E B2RXH2 1/20 0.33
PDE5A O76074 1/20 0.33
TNF P01375 1/20 0.33
MAPK1 P28482 1/20 0.33
BLM P54132 1/20 0.33
PDE1A P54750 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11206098 1.00 MAPT (0.38) MAPTMAP3K14PDE4APDE4BPDE4C
SCHEMBL13977388 1.00 MAPT (0.38) MAPTMAP3K14PDE4APDE4BPDE4C
SCHEMBL11206101 1.00 MAPT (0.38) MAPTMAP3K14PDE4APDE4BPDE4C
SCHEMBL20343542 0.95 MAP3K14 (0.34) MAPTMAP3K14MTNR1APKM
SCHEMBL7217095 0.93 ALDH1A1 (0.40) MAPTMAP3K14PDE4APDE4BPDE4C
SCHEMBL2380603 0.91 ALDH1A1 (0.38) MAPTMAP3K14PDE4APDE4BPDE4C
SCHEMBL7794999 0.90
SCHEMBL7214892 0.88 MAP3K14 (0.36) MAPTMAP3K14PDE4APDE4BPDE4C
SCHEMBL25175873 0.83 SLC6A1 (0.35) MAPTMAP3K14LMNAKDM4EKMT2A
SCHEMBL26984265 0.82

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0090362-A2 Derivatives of cycloalka(c)pyrrole-carboxylic acids, process for their preparation, agents containing them and their use, as well as cycloalka(c)pyrrole-carboxylic acids as intermediates, and process for their preparation HOECHST AKTIENGESELLSCHAFT (DE) 1983-10-05 EP disclosed