SCHEMBL11207874

SCHEMBL11207874

C[C@H]1OC(O)C[C@H](O)[C@@H]1O.C[C@H]1OC(O)C[C@H](O)[C@@H]1O.C[C@]1(O)CC[C@]2(C)C3CC[C@@]4(C)C(CC[C@@H]4C4=CC(=O)OC4)C3CC[C@@H]2C1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATP1A1 P05023 8/20 0.52
ATP1B1 P05026 8/20 0.52
ATP1A3 P13637 8/20 0.52
ATP1B2 P14415 8/20 0.52
ATP1A2 P50993 8/20 0.52
ATP1B3 P54709 8/20 0.52
FXYD2 P54710 8/20 0.52
ATP1A4 Q13733 8/20 0.52
TP53 P04637 8/20 0.50
SMN1; SMN2 Q16637 6/20 0.50
LMNA P02545 6/20 0.50
RAB9A P51151 4/20 0.50
NPC1 O15118 3/20 0.50
STAT3 P40763 2/20 0.50
USP2 O75604 1/20 0.50
ABCB11 O95342 1/20 0.50
MAPT P10636 1/20 0.50
SLCO4C1 Q6ZQN7 1/20 0.50
PAX8 Q06710 3/20 0.48
HIF1A Q16665 3/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8830484 0.89 TP53 (0.56) ATP1A1ATP1B1ATP1A3ATP1B2ATP1A2
SCHEMBL8830696 0.89 TP53 (0.56) ATP1A1ATP1B1ATP1A3ATP1B2ATP1A2
SCHEMBL11211273 0.88 ATP1A1 (0.53) ATP1A1ATP1B1ATP1A3ATP1B2ATP1A2
SCHEMBL11208371 0.88 ATP1A1 (0.52) ATP1A1ATP1B1ATP1A3ATP1B2ATP1A2
SCHEMBL9762798 0.82 ATP1A1 (0.52) ATP1A1ATP1B1ATP1A3ATP1B2ATP1A2
Ethyl Acetate SCHEMBL2958120 0.82 ATP1A1 (0.51) ATP1A1ATP1B1ATP1A3ATP1B2ATP1A2
Ethyl Acetate SCHEMBL2960997 0.81 ATP1A1 (0.50) ATP1A1ATP1B1ATP1A3ATP1B2ATP1A2
SCHEMBL3374210 0.80 ATP1A1 (0.75) ATP1A1ATP1B1ATP1A3ATP1B2ATP1A2
SCHEMBL8190252 0.79 ATP1A1 (0.50) ATP1A1ATP1B1ATP1A3ATP1B2ATP1A2
SCHEMBL11208403 0.78 TP53 (0.54) ATP1A1ATP1B1ATP1A3ATP1B2ATP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0047928-B1 CARDENOLIDE-BIS-DIGITOXOSIDE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR UTILIZATION AS MEDICINES Roche Diagnostics GmbH (DE) 1983-09-21 EP disclosed
US-4353895-A CARDIOTONIC AGENTS WITH DESIRABLE RATES OF EXCRETION, PRIMARILY EXTRARENALLY BOEHRINGER MANNHEIM GMBH (DE) 1982-10-12 US disclosed
EP-0047928-A1 Cardenolide-bis-digitoxoside derivatives, process for their preparation and their utilization as medicines Roche Diagnostics GmbH (DE) 1982-03-24 EP disclosed