SCHEMBL11207914

SCHEMBL11207914

O=CNc1cccc(NC=O)c1O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.44
KDM5A P29375 2/20 0.42
PABPC1 P11940 1/20 0.42
ALDH1A1 P00352 2/20 0.42
ERN1 O75460 4/20 0.38
RXFP1 Q9HBX9 1/20 0.37
ADAMTS4 O75173 1/20 0.33
EGFR P00533 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
LMNA P02545 1/20 0.33
FYN P06241 1/20 0.33
MMP2 P08253 1/20 0.33
MMP9 P14780 1/20 0.33
HPGD P15428 1/20 0.33
ALOX15 P16050 1/20 0.33
MMP8 P22894 1/20 0.33
CA6 P23280 1/20 0.33
CDK2 P24941 1/20 0.33
MMP12 P39900 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3567350 0.89 ERN1 (0.48) TSHRKDM5APABPC1ALDH1A1ERN1
SCHEMBL14625516 0.85 KDM5A (0.41) TSHRKDM5APABPC1ALDH1A1LMNA
SCHEMBL3730357 0.85 ERN1 (0.55) TSHRKDM5APABPC1ALDH1A1ERN1
SCHEMBL13412750 0.85 ALDH1A1 (0.50) TSHRKDM5APABPC1ALDH1A1LMNA
SCHEMBL4297093 0.82 ALDH1A1 (0.51) KDM5AALDH1A1RXFP1CA1CA2
SCHEMBL3730352 0.82 CXCR2 (0.40) TSHRKDM5APABPC1ALDH1A1ERN1
SCHEMBL14458133 0.80 RXFP1 (0.43) KDM5AALDH1A1RXFP1LMNAHPGD
SCHEMBL1765338 0.80 CXCR2 (0.50) TSHRALDH1A1ERN1RXFP1LMNA
SCHEMBL31486082 0.80 CXCR2 (0.50) TSHRALDH1A1ERN1RXFP1LMNA
SCHEMBL14475281 0.80 RXFP1 (0.43) KDM5AALDH1A1RXFP1LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0022387-B1 PROCESS FOR THE PREPARATION OF BENZENE DERIVATIVES BY THE REACTION OF AN ACTIVATED HALOBENZENE WITH AN ORGANIC COMPOUND CONTAINING AN OXYGEN OR SULPHUR ANION RHONE-POULENC SPECIALITES CHIMIQUES (FR) 1983-01-05 EP disclosed
EP-0022387-A1 Process for the preparation of benzene derivatives by the reaction of an activated halobenzene with an organic compound containing an oxygen or sulphur anion RHONE-POULENC SPECIALITES CHIMIQUES (FR) 1981-01-14 EP disclosed