SCHEMBL11209183

SCHEMBL11209183

COc1ccc(C2=c3cc4c(cc3N(C(C)=O)C2=O)=C(c2ccccc2)C(=O)O4)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 4/20 0.39
NR1H3 Q13133 4/20 0.39
MEN1 O00255 1/20 0.38
USP2 O75604 1/20 0.38
MAPT P10636 1/20 0.38
CASP1 P29466 1/20 0.38
BRCA1 P38398 1/20 0.38
KMT2A Q03164 1/20 0.38
BACE1 P56817 3/20 0.37
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
MAOB P27338 1/20 0.36
GABRA1 P14867 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
GABRA2 P47869 1/20 0.35
FGFR1 P11362 1/20 0.35
SRC P12931 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11364695 0.97 MAPT (0.38) NR1H2NR1H3MEN1USP2MAPT
SCHEMBL11214857 0.91 MAPT (0.41) MEN1USP2MAPTCASP1BRCA1
SCHEMBL11368447 0.84 MAPT (0.40) MEN1USP2MAPTCASP1BRCA1
SCHEMBL8089080 0.82 BACE1 (0.47) NR1H2NR1H3MEN1MAPTKMT2A
SCHEMBL11363941 0.82 NR1H2 (0.42) NR1H2NR1H3MEN1MAPTKMT2A
SCHEMBL17432753 0.79 ME2 (0.47) MEN1MAPTKMT2ABACE1
SCHEMBL11215197 0.76 KMT2A (0.42) NR1H2NR1H3MEN1USP2MAPT
SCHEMBL11206044 0.76 NR1H2 (0.40) NR1H2NR1H3MAPT
SCHEMBL11211990 0.76 MEN1 (0.35) MEN1USP2MAPTCASP1BRCA1
SCHEMBL17430475 0.74 ALKBH3 (0.47) MEN1MAPTKMT2AMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0033583-B1 DYESTUFFS COMPRISING TWO 5-MEMBERED HETEROCYCLIC NUCLEI FUSED TO A CENTRAL CYCLOHEXADIENE NUCLEUS, PROCESSES FOR THEIR PREPARATION AND THEIR USE FOR COLOURING SYNTHETIC TEXTILE MATERIALS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1983-10-12 EP disclosed
EP-0033583-A1 Dyestuffs comprising two 5-membered heterocyclic nuclei fused to a central cyclohexadiene nucleus, processes for their preparation and their use for colouring synthetic textile materials IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1981-08-12 EP disclosed