SCHEMBL11209491

SCHEMBL11209491

C=CCc1c(CC(=O)N(CCC)CCC)ccc(OC)c1OC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
TSHR P16473 1/20 0.42
APP P05067 2/20 0.39
POLB P06746 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
APEX1 P27695 1/20 0.37
PTGS1 P23219 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 1/20 0.36
HPGD P15428 1/20 0.36
ALOX5 P09917 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.34
LMNA P02545 1/20 0.34
PPARG P37231 1/20 0.34
PPARD Q03181 1/20 0.34
PPARA Q07869 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11213474 0.81 HSD17B10 (0.47) CYP3A4POLBTDP1PTGS1NPSR1
Ammonia Solution, Strong SCHEMBL10969833 0.78 ALDH1A1 (0.44) CYP3A4POLBTDP1PTGS1ALDH1A1
SCHEMBL11210388 0.78 AOC3 (0.43) POLBAOC3
SCHEMBL11025102 0.72 POLB (0.44) CYP3A4POLBTDP1PTGS1ALDH1A1
SCHEMBL10969347 0.71 POLB (0.43) CYP3A4POLBPTGS1ALDH1A1KDM4E
SCHEMBL10536230 0.71 PTGS1 (0.62) CYP3A4TSHRPOLBTDP1PTGS1
SCHEMBL11553227 0.70 CYP3A4 (0.45) CYP3A4TSHRPOLBTDP1PTGS1
SCHEMBL6430390 0.70 TDP1 (0.55) CYP3A4POLBTDP1PTGS1ALDH1A1
SCHEMBL10970024 0.70 TAAR1 (0.44) CYP3A4CYP1A2POLBALDH1A1KDM4E
SCHEMBL28626652 0.69 MAPT (0.43) CYP3A4POLBTDP1PTGS1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0036773-B1 2,3-DIHYDROBENZOFURANS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SMITHKLINE BECKMAN CORPORATION (US) 1983-02-16 EP disclosed
EP-0036773-A1 2,3-Dihydrobenzofurans, process for their preparation and pharmaceutical compositions containing them SMITHKLINE BECKMAN CORPORATION (US) 1981-09-30 EP disclosed
US-4254140-A USED FOR CARDIOVASCULAR DISORDERS; HYPOTENSIVE AGENT SMITHKLINE CORPORATION (US) 1981-03-03 US disclosed