SCHEMBL11211642

SCHEMBL11211642

CCC(NC(=O)O)C1CCCCC1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 3/20 0.46
SHBG P04278 1/20 0.43
CA12 O43570 2/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
MMP2 P08253 2/20 0.40
CA9 Q16790 2/20 0.40
TSHR P16473 2/20 0.39
ALDH1A1 P00352 3/20 0.38
NPSR1 Q6W5P4 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
KDM4E B2RXH2 1/20 0.37
P2RX7 Q99572 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
THRB P10828 1/20 0.37
ATM Q13315 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5510787 0.85 SMN1; SMN2 (0.45) EPHX1SHBGCA12CA1CA2
SCHEMBL14277937 0.85 EPHX1 (0.46) EPHX1SHBGCA12CA1CA2
SCHEMBL13274039 0.83 EPHX1 (0.45) EPHX1SHBGCA12CA1CA2
SCHEMBL8078353 0.83 EPHX1 (0.45) EPHX1SHBGCA12CA1CA2
SCHEMBL25297559 0.82 P2RX7 (0.47) EPHX1CA12CA1CA2MMP2
SCHEMBL15909256 0.82 P2RX7 (0.47) EPHX1CA12CA1CA2MMP2
SCHEMBL25297558 0.82 P2RX7 (0.47) EPHX1CA12CA1CA2MMP2
SCHEMBL22233331 0.81 CPN1 (0.50) EPHX1TSHRSMN1; SMN2KDM4EL3MBTL1
SCHEMBL20774033 0.81 DPP4 (0.51) EPHX1CA12CA1CA2MMP2
SCHEMBL22341347 0.81 ALDH1A1 (0.38) EPHX1CA12CA1CA2MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012098065-A1 PYRIDO PYRIMIDINES FOR USE AS DYRK1 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2012-07-26 WO disclosed
US-4360633-A Coating solution of polyetherimide oligomers GENERAL ELECTRIC COMPANY (US) 1982-11-23 US disclosed
EP-0017772-B1 METHOD OF IMPROVING THE SOLUBILITY OF BIOLOGICALLY ACTIVE AGENTS IN WATER AND IN LOWER ALIPHATIC ALCOHOLS, AND COMPOUNDS HAVING AN IMPROVED SOLUBILITY BAYER AG (DE) 1982-07-28 EP disclosed
EP-0014263-B1 METHOD OF IMPROVING THE SOLUBILITY OF BIOLOGICALLY ACTIVE AGENTS IN WATER AND IN LOWER ALIPHATIC ALCOHOLS, AND COMPOUNDS HAVING AN IMPROVED SOLUBILITY BAYER AG (DE) 1982-05-05 EP disclosed
EP-0017772-A1 Method of improving the solubility of biologically active agents in water and in lower aliphatic alcohols, and compounds having an improved solubility BAYER AG (DE) 1980-10-29 EP disclosed
EP-0014263-A2 Method of improving the solubility of biologically active agents in water and in lower aliphatic alcohols, and compounds having an improved solubility BAYER AG (DE) 1980-08-20 EP disclosed