SCHEMBL11212923

SCHEMBL11212923

COc1ccc2c(c1)CC[C@@H]1[C@@H]2CC[C@]2(C)C(=O)[C@H](OC(C)=O)C[C@@H]12

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.67
LMNA P02545 6/20 0.63
HSD17B1 P14061 5/20 0.63
SMN1; SMN2 Q16637 3/20 0.63
MAPT P10636 2/20 0.63
RECQL P46063 2/20 0.63
HSD17B10 Q99714 1/20 0.57
CYP3A4 P08684 4/20 0.56
TP53 P04637 1/20 0.56
PGR P06401 2/20 0.53
SLC6A3 Q01959 2/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2C19 P33261 1/20 0.53
HIF1A Q16665 1/20 0.53
NR3C1 P04150 1/20 0.53
CNR1 P21554 1/20 0.53
SLC6A2 P23975 1/20 0.53
SLC6A4 P31645 1/20 0.53
ADORA3 P0DMS8 1/20 0.53
AR P10275 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11209381 0.92 SMN1; SMN2 (0.67) ESR1LMNAHSD17B1SMN1; SMN2MAPT
SCHEMBL351004 0.92 SMN1; SMN2 (0.67) ESR1LMNAHSD17B1SMN1; SMN2MAPT
SCHEMBL351005 0.92 SMN1; SMN2 (0.67) ESR1LMNAHSD17B1SMN1; SMN2MAPT
SCHEMBL8042918 0.88 ESR1 (0.73) ESR1LMNAHSD17B1SMN1; SMN2MAPT
SCHEMBL7518036 0.86 MAPT (0.63) ESR1LMNAHSD17B1SMN1; SMN2MAPT
SCHEMBL11865928 0.85 ESR1 (0.74) ESR1LMNAHSD17B1SMN1; SMN2MAPT
SCHEMBL15979565 0.83 HSD17B1 (0.71) ESR1LMNAHSD17B1SMN1; SMN2MAPT
SCHEMBL11231177 0.83 HSD17B1 (0.71) ESR1LMNAHSD17B1SMN1; SMN2MAPT
SCHEMBL309293 0.83 HSD17B1 (0.69) ESR1LMNAHSD17B1SMN1; SMN2MAPT
SCHEMBL9558249 0.83 LMNA (0.69) ESR1LMNAHSD17B1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0033561-B1 NOVEL 17-AMINO-16-HYDROXY STEROIDS OF THE ANDROSTANE AND OESTRANE SERIES AND DERIVATIVES THEREOF, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS AKZO N.V. (NL) 1983-05-11 EP disclosed
US-4330539-A Novel 17-amino-16-hydroxy steroids of the androstane and oestrane series and derivatives thereof AKZO NV (NL) 1982-05-18 US disclosed
US-4298538-A 16-Dimethylaminomethylene-3-methoxy-1,3,5-(10)-estratrien-17-one, a process for the preparation thereof and its use as a preparative intermediate SCHERING, AKTIENGESELLSCHAFT (DE) 1981-11-03 US disclosed
EP-0033561-A1 Novel 17-amino-16-hydroxy steroids of the androstane and oestrane series and derivatives thereof, processes for their preparation and pharmaceutical compositions AKZO N.V. (NL) 1981-08-12 EP disclosed