SCHEMBL11213690

SCHEMBL11213690

CN[C@H]1[C@H](O)C[C@H]2[C@@H]3CCc4cc(OC(C)=O)ccc4[C@H]3CC[C@@]21C

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 6/20 0.69
LMNA P02545 4/20 0.69
SMN1; SMN2 Q16637 3/20 0.69
ATM Q13315 3/20 0.69
PGR P06401 2/20 0.69
AR P10275 2/20 0.69
SLC6A3 Q01959 2/20 0.69
ADORA3 P0DMS8 2/20 0.69
CHRM1 P11229 1/20 0.69
TBXA2R P21731 1/20 0.69
ADRA1A P35348 1/20 0.69
OPRM1 P35372 1/20 0.69
MAPT P10636 3/20 0.65
TP53 P04637 1/20 0.65
CYP3A4 P08684 1/20 0.65
ESR2 Q92731 2/20 0.55
NR3C1 P04150 2/20 0.55
SHBG P04278 2/20 0.55
SLC6A4 P31645 2/20 0.55
CYP2C9 P11712 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Maleic Acid SCHEMBL11229073 0.95 ESR1 (0.63) ESR1LMNASMN1; SMN2ATMPGR
SCHEMBL11209403 0.91 ESR1 (0.57) ESR1LMNASMN1; SMN2ATMPGR
SCHEMBL11207655 0.90 MAPT (0.66) ESR1LMNASMN1; SMN2ATMPGR
SCHEMBL5529984 0.89 ESR1 (0.76) ESR1LMNASMN1; SMN2ATMPGR
SCHEMBL2518701 0.89 ESR1 (0.76) ESR1LMNASMN1; SMN2ATMPGR
SCHEMBL23037707 0.89 ESR1 (0.76) ESR1LMNASMN1; SMN2ATMPGR
SCHEMBL21523191 0.89 ESR1 (0.76) ESR1LMNASMN1; SMN2ATMPGR
SCHEMBL11214603 0.88 LMNA (0.67) ESR1LMNASMN1; SMN2ATMPGR
SCHEMBL11216046 0.88 LMNA (0.67) ESR1LMNASMN1; SMN2ATMPGR
SCHEMBL11219023 0.88 LMNA (0.67) ESR1LMNASMN1; SMN2ATMPGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0033561-B1 NOVEL 17-AMINO-16-HYDROXY STEROIDS OF THE ANDROSTANE AND OESTRANE SERIES AND DERIVATIVES THEREOF, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS AKZO N.V. (NL) 1983-05-11 EP disclosed
US-4330539-A Novel 17-amino-16-hydroxy steroids of the androstane and oestrane series and derivatives thereof AKZO NV (NL) 1982-05-18 US disclosed
EP-0033561-A1 Novel 17-amino-16-hydroxy steroids of the androstane and oestrane series and derivatives thereof, processes for their preparation and pharmaceutical compositions AKZO N.V. (NL) 1981-08-12 EP disclosed