SCHEMBL1121608

SCHEMBL1121608

O=C(NCCO)c1cccc2oc(NC3CCNCC3)nc12

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 12/20 0.43
KCNH2 Q12809 2/20 0.41
CYP2C19 P33261 1/20 0.41
PARP1 P09874 2/20 0.40
AURKA O14965 1/20 0.39
RPS6KB1 P23443 1/20 0.39
CHRM1 P11229 3/20 0.37
PBK Q96KB5 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1121676 0.85 HTR3A (0.42) HTR3AKCNH2CYP2C19PARP1AURKA
SCHEMBL4155160 0.83 RPS6KB1 (0.43) HTR3AKCNH2CYP2C19PARP1AURKA
SCHEMBL1121563 0.81 RIPK1 (0.48) HTR3AKCNH2CYP2C19PARP1AURKA
SCHEMBL1121750 0.80 PARP1 (0.47) HTR3APARP1CHRM1
SCHEMBL1121260 0.78 POLB (0.43) HTR3A
SCHEMBL1121610 0.78 RPS6KB1 (0.41) HTR3APARP1AURKARPS6KB1
SCHEMBL1121178 0.74 SSTR5 (0.64) KCNH2
SCHEMBL1121350 0.74 IRAK4 (0.36) AURKARPS6KB1
SCHEMBL1121250 0.73 SSTR5 (0.65) KCNH2
SCHEMBL1121464 0.72 SSTR5 (0.57) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924579-B1 BENZOOXAZOLE, OXAZOLOPYRIDINE, BENZOTHIAZOLE AND THIAZOLOPYRIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2011-02-09 EP disclosed