SCHEMBL11220107

SCHEMBL11220107

COc1cc2c(cc1OC)C(CC(C)(C)CBr)(c1ccc(F)cc1)OCCC2

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.35
TMEM97 Q5BJF2 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
KMT2A Q03164 2/20 0.33
MAOB P27338 1/20 0.33
ABCB1 P08183 2/20 0.32
SLC6A4 P31645 2/20 0.31
ACHE P22303 1/20 0.31
KDM4C Q9H3R0 1/20 0.31
BCHE P06276 1/20 0.31
MEN1 O00255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11221675 0.81 SLC6A4 (0.39) KCNH2SIGMAR1SLC6A4ACHEBCHE
SCHEMBL11226959 0.81 SLC6A4 (0.33) KCNH2SIGMAR1SLC6A4ACHE
SCHEMBL11223876 0.79 ALDH1A1 (0.32)
SCHEMBL11225546 0.79 SLC6A4 (0.41) KCNH2SIGMAR1SLC6A4ACHEBCHE
SCHEMBL11220962 0.78 SLC6A4 (0.40) KCNH2SIGMAR1SLC6A4ACHEBCHE
SCHEMBL11220849 0.77 KCNH2 (0.35) KCNH2TMEM97SIGMAR1KMT2AMAOB
SCHEMBL11222322 0.76 SLC6A4 (0.40) KCNH2SIGMAR1SLC6A4ACHEBCHE
SCHEMBL11224396 0.73 SLC6A4 (0.41) KCNH2SIGMAR1SLC6A4ACHEBCHE
SCHEMBL11223955 0.72 SLC6A4 (0.41) KCNH2SIGMAR1SLC6A4ACHEBCHE
SCHEMBL11222621 0.72 TACR1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4352805-A BENZOXEPINE DERIVATIVES THE UPJOHN COMPANY (US) 1982-10-05 US disclosed
US-4251526-A HYPOTENSIVE AGENTS AND ANTIPSYCHOTIC PHARMACIA & UPJOHN COMPANY 1981-02-17 US disclosed
US-4250175-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS PHARMACIA & UPJOHN COMPANY 1981-02-10 US disclosed
US-4250181-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1981-02-10 US disclosed
US-4247553-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1981-01-27 US disclosed
US-4179510-A ISOCHROMANS AND 2-BENZOXEPINS THE UPJOHN COMPANY (US) 1979-12-18 US disclosed
US-4153612-A 2-Benzoxepins THE UPJOHN COMPANY (US) 1979-05-08 US disclosed