SCHEMBL11220193

SCHEMBL11220193

COc1ccc(CC(C)(C)S)cc1OC

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.59
CYP19A1 P11511 1/20 0.53
ATM Q13315 2/20 0.52
KDM4E B2RXH2 1/20 0.52
ALDH1A1 P00352 2/20 0.50
PPARG P37231 1/20 0.50
PPARD Q03181 1/20 0.50
PPARA Q07869 1/20 0.50
POLB P06746 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
BLM P54132 1/20 0.47
PMP22 Q01453 1/20 0.47
AOC3 Q16853 1/20 0.46
LDHA P00338 1/20 0.46
SIGMAR1 Q99720 1/20 0.45
STAT3 P40763 1/20 0.45
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL74008 0.84 CA2 (0.63) CA2CYP19A1ATMKDM4EALDH1A1
SCHEMBL5114730 0.82 CA2 (0.61) CA2CYP19A1ATMKDM4EALDH1A1
SCHEMBL11220959 0.81 CA2 (0.55) CA2CYP19A1ATMKDM4EALDH1A1
SCHEMBL11258047 0.81 CA2 (0.59) CA2CYP19A1ATMKDM4EALDH1A1
SCHEMBL10730478 0.81 CA2 (0.59) CA2CYP19A1ATMKDM4EALDH1A1
SCHEMBL5114907 0.81 CA2 (0.59) CA2CYP19A1ATMKDM4EALDH1A1
Hydrochloric Acid SCHEMBL11329627 0.79 CA2 (0.57) CA2CYP19A1ATMKDM4EALDH1A1
SCHEMBL13509578 0.79 CA2 (0.57) CA2CYP19A1ATMKDM4EALDH1A1
SCHEMBL13144840 0.79 CA2 (0.57) CA2CYP19A1ATMKDM4EALDH1A1
SCHEMBL29944152 0.79 CA2 (0.57) CA2CYP19A1ATMKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4352805-A BENZOXEPINE DERIVATIVES THE UPJOHN COMPANY (US) 1982-10-05 US disclosed
US-4312868-A HYPOTENSIVE, ANTIPSYCHOTIC THE UPJOHN COMPANY (US) 1982-01-26 US disclosed
US-4251526-A HYPOTENSIVE AGENTS AND ANTIPSYCHOTIC PHARMACIA & UPJOHN COMPANY 1981-02-17 US disclosed
US-4250175-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS PHARMACIA & UPJOHN COMPANY 1981-02-10 US disclosed
US-4250181-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1981-02-10 US disclosed
US-4247553-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1981-01-27 US disclosed
US-4179510-A ISOCHROMANS AND 2-BENZOXEPINS THE UPJOHN COMPANY (US) 1979-12-18 US disclosed
US-4166062-A HYPOTENSIVE AGENTS, CNS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1979-08-28 US disclosed
US-4153612-A 2-Benzoxepins THE UPJOHN COMPANY (US) 1979-05-08 US disclosed