SCHEMBL112235

SCHEMBL112235

COc1ccc(-c2nc(C(=O)N3CCN(c4ccccc4C(=O)Nc4cccnc4)CC3)cs2)cc1OC.O=C(Nc1cccnc1)c1ccccc1N1CCN(C(=O)Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)CC1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 4/20 0.47
ALDH1A1 P00352 1/20 0.42
TLR7 Q9NYK1 1/20 0.41
TP53 P04637 2/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
MAPT P10636 3/20 0.40
KDM4E B2RXH2 2/20 0.40
LMNA P02545 1/20 0.40
IRAK4 Q9NWZ3 4/20 0.40
LRRK2 Q5S007 1/20 0.39
TRPV1 Q8NER1 1/20 0.39
IDE P14735 1/20 0.39
MAPK1 P28482 1/20 0.39
MAPK10 P53779 1/20 0.39
HTR7 P34969 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL113391 0.90 CHEK1 (0.54) CHEK1ALDH1A1TLR7TP53NPC1
SCHEMBL111521 0.83 TRPV1 (0.54) ALDH1A1MAPTKDM4ELMNALRRK2
SCHEMBL13075778 0.73 ALDH1A1 (0.49) ALDH1A1TP53NPC1RAB9AMAPT
SCHEMBL115046 0.72 LMNA (0.58) ALDH1A1TP53NPC1RAB9AMAPT
SCHEMBL112384 0.69 GAA (0.52) NPC1RAB9AMAPTKDM4ELMNA
SCHEMBL113246 0.68 GAA (0.52) NPC1RAB9AMAPTKDM4ELMNA
SCHEMBL111258 0.68 LMNA (0.51) ALDH1A1NPC1RAB9AMAPTKDM4E
SCHEMBL113253 0.67 LMNA (0.57) ALDH1A1TP53NPC1RAB9AMAPT
SCHEMBL112552 0.67 LMNA (0.57) ALDH1A1TP53NPC1RAB9AMAPT
SCHEMBL111089 0.67 POLB (0.63) ALDH1A1TP53NPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2424858-A1 CXCR3 RECEPTOR ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2012-03-07 EP disclosed