SCHEMBL11223697

SCHEMBL11223697

COC(=O)C1CSCN1C(=O)C(C)O

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACE P12821 2/20 0.47
NPSR1 Q6W5P4 1/20 0.46
HSD17B10 Q99714 1/20 0.46
DPP4 P27487 3/20 0.37
DPP8 Q6V1X1 2/20 0.37
DPP7 Q9UHL4 2/20 0.37
PEPD P12955 5/20 0.36
XPNPEP1 Q9NQW7 2/20 0.36
MMP2 P08253 2/20 0.34
ANPEP P15144 2/20 0.34
PREP P48147 1/20 0.32
CYP1A2 P05177 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27970159 0.86 ACE (0.46) ACENPSR1HSD17B10DPP4DPP8
SCHEMBL11342331 0.81 HSD17B10 (0.51) ACENPSR1HSD17B10MMP2ANPEP
SCHEMBL9109446 0.80 NPSR1 (0.50) ACENPSR1HSD17B10DPP4DPP8
SCHEMBL11155540 0.79 ACE (0.49) ACENPSR1HSD17B10DPP4DPP8
SCHEMBL11164632 0.78 ACE (0.48) ACENPSR1HSD17B10DPP4DPP8
SCHEMBL11355229 0.78 ACE (0.48) ACENPSR1HSD17B10
SCHEMBL200924 0.76 RAB9A (0.46) ACENPSR1HSD17B10DPP4DPP8
SCHEMBL27970157 0.74 NPSR1 (0.46) ACENPSR1HSD17B10DPP4DPP8
SCHEMBL27970090 0.73 HSD17B10 (0.45) ACENPSR1HSD17B10DPP4DPP8
SCHEMBL200923 0.73 ATM (0.46) NPSR1HSD17B10DPP4DPP8DPP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4316896-A Aminoacid derivatives as antihypertensives MERCK & CO., INC. (US) 1982-02-23 US disclosed
EP-0009183-B1 PHOSPHORYL AMINOACID DERIVATIVES AND COMPOSITION FOR TREATING HYPERTENSION CONTAINING THE SAME MERCK & CO. INC. (US) 1981-10-21 EP disclosed
EP-0009183-A1 Phosphoryl aminoacid derivatives and composition for treating hypertension containing the same MERCK & CO. INC. (US) 1980-04-02 EP disclosed