SCHEMBL11223992

SCHEMBL11223992

CC(=O)Nc1cc(-c2ccnc(C)c2C)ccc1[N+](=O)[O-]

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
NPSR1 Q6W5P4 2/20 0.42
POLB P06746 2/20 0.42
PIK3C3 Q8NEB9 2/20 0.42
HPGD P15428 2/20 0.42
GALR2 O43603 1/20 0.42
MITF O75030 1/20 0.42
LMNA P02545 1/20 0.42
HSP90AA1 P07900 1/20 0.42
XBP1 P17861 1/20 0.42
CCR6 P51684 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MAPT P10636 2/20 0.41
PKM P14618 2/20 0.41
TOP2A P11388 4/20 0.40
KMT2A Q03164 2/20 0.40
MAPK1 P28482 1/20 0.40
HTT P42858 1/20 0.40
TDP1 Q9NUW8 1/20 0.38
PDE7A Q13946 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11225695 0.83 PIK3C3 (0.48) ALDH1A1NPSR1POLBPIK3C3HPGD
SCHEMBL11375763 0.80 MAPT (0.49) ALDH1A1NPSR1POLBHPGDLMNA
SCHEMBL11233932 0.77 HDAC1 (0.48) NPSR1POLBMAPTKMT2AHTT
SCHEMBL11224373 0.77 MAPT (0.47) ALDH1A1NPSR1POLBHPGDGALR2
SCHEMBL11224469 0.77 PIK3C3 (0.44) ALDH1A1NPSR1POLBPIK3C3HPGD
SCHEMBL11220980 0.76 KMT2A (0.43) ALDH1A1NPSR1POLBPIK3C3HPGD
SCHEMBL11277648 0.74 MAPT (0.53) NPSR1POLBPIK3C3MAPTPKM
SCHEMBL22535975 0.73 CYP3A4 (0.55) ALDH1A1NPSR1POLBHPGDGALR2
SCHEMBL11224541 0.73 ABCB1 (0.54) ALDH1A1HPGDMAPTKMT2AABCB1
SCHEMBL11222535 0.72 PIK3C3 (0.55) ALDH1A1POLBPIK3C3LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0056260-A1 Pyridinyl-substituted-benz imidazole derivatives and preparation STERLING DRUG INC. (US) 1982-07-21 EP disclosed
EP-0055453-A2 5-(Pyridinyl)-benzimidazole derivatives and preparation STERLING DRUG INC. (US) 1982-07-07 EP disclosed
US-4335132-A 5-(Py-Y)-1H-benzimidazol-2-ols and 5-(Py-Y-)-1H-benzimidazole-2-thiols STERLING DRUG, INC. (US) 1982-06-15 US disclosed
US-4331671-A 5-(Pyridinyl)-1H-benzimidazoles and 1-hydroxy-6-(pyridinyl)-1H-benzimidazoles and their cardiotonic use STERLING DRUG INC. (US) 1982-05-25 US disclosed