SCHEMBL11224064

SCHEMBL11224064

COc1cc2c(cc1Br)C(CCCl)OCC2

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 9/20 0.45
HTR2A P28223 7/20 0.45
HTR2B P41595 6/20 0.45
ALDH1A1 P00352 1/20 0.37
TAAR1 Q96RJ0 1/20 0.37
CYP19A1 P11511 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11220870 0.92 HTR2C (0.43) HTR2CHTR2AHTR2BCYP19A1
SCHEMBL9688216 0.89 KCNN2 (0.43) ALDH1A1TAAR1
SCHEMBL11224510 0.85 HTR2C (0.48) HTR2CHTR2AHTR2BALDH1A1TAAR1
SCHEMBL11222930 0.82 HTR2A (0.47) HTR2CHTR2AHTR2BALDH1A1TAAR1
SCHEMBL10990476 0.81 KCNN2 (0.41) ALDH1A1
SCHEMBL11370362 0.81 KCNN2 (0.41) ALDH1A1
SCHEMBL11220460 0.81 KCNN2 (0.44) ALDH1A1TAAR1
SCHEMBL11217845 0.80 KCNN2 (0.43) ALDH1A1TAAR1
SCHEMBL11222512 0.78 HTR2C (0.40) HTR2CHTR2AHTR2BALDH1A1TAAR1
SCHEMBL7290833 0.77 ALDH1A1 (0.43) ALDH1A1TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4352805-A BENZOXEPINE DERIVATIVES THE UPJOHN COMPANY (US) 1982-10-05 US disclosed
US-4312868-A HYPOTENSIVE, ANTIPSYCHOTIC THE UPJOHN COMPANY (US) 1982-01-26 US disclosed
US-4251526-A HYPOTENSIVE AGENTS AND ANTIPSYCHOTIC PHARMACIA & UPJOHN COMPANY 1981-02-17 US disclosed
US-4250181-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1981-02-10 US disclosed
US-4250175-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS PHARMACIA & UPJOHN COMPANY 1981-02-10 US disclosed
US-4247553-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1981-01-27 US disclosed
US-4179510-A ISOCHROMANS AND 2-BENZOXEPINS THE UPJOHN COMPANY (US) 1979-12-18 US disclosed
US-4166062-A HYPOTENSIVE AGENTS, CNS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1979-08-28 US disclosed
US-4153612-A 2-Benzoxepins THE UPJOHN COMPANY (US) 1979-05-08 US disclosed