SCHEMBL11224196

SCHEMBL11224196

Clc1ccc2c(c1)OC(CCBr)CO2

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.56
CA1 P00915 1/20 0.49
FFAR1 O14842 12/20 0.43
MAPT P10636 1/20 0.42
HBB P68871 1/20 0.42
HTR1A P08908 1/20 0.42
DRD2 P14416 1/20 0.42
DRD4 P21917 1/20 0.42
ADRA1D P25100 1/20 0.42
HTR2C P28335 1/20 0.42
ADRA1A P35348 1/20 0.42
ADRA1B P35368 1/20 0.42
DRD3 P35462 1/20 0.42
CYP2C9 P11712 1/20 0.40
CYP2B6 P20813 1/20 0.40
SLCO1B3 Q9NPD5 1/20 0.40
HTT P42858 1/20 0.40
MTNR1A P48039 1/20 0.40
NPC1 O15118 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11230966 0.94 CA2 (0.56) CA2CA1FFAR1MAPTHBB
SCHEMBL15864967 0.87 CA2 (0.58) CA2CA1FFAR1HTR1ADRD2
SCHEMBL15864969 0.87 CA2 (0.58) CA2CA1FFAR1HTR1ADRD2
SCHEMBL6761878 0.84 CA2 (0.59) CA2CA1FFAR1MAPTHBB
SCHEMBL11025999 0.82 CA2 (0.59) CA2CA1FFAR1HTR1ADRD2
SCHEMBL11235851 0.81 CA2 (0.56) CA2FFAR1MAPTHTTMTNR1A
SCHEMBL16089590 0.81 CA2 (0.58) CA2CA1FFAR1HTR1ADRD2
SCHEMBL440872 0.81 CA2 (0.62) CA2CA1FFAR1HTR1ADRD2
SCHEMBL1044791 0.81 CA2 (0.58) CA2CA1FFAR1MAPTHBB
SCHEMBL4764921 0.81 CA2 (0.62) CA2CA1FFAR1HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4353901-A HYPERTENSION, CONGESTIVE HEART FAILURE, ARRHYTHMIAMIGRAINE, VASOSPASTIC DISORDERS, ASTHMA SYNTEX (U.S.A.) INC. (US) 1982-10-12 US disclosed