SCHEMBL11224271

SCHEMBL11224271

COc1ccc2c(c1OC)C(CBr)SCC(C1CCCC1)C2

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.36
NQO2 P16083 1/20 0.34
MTNR1A P48039 1/20 0.34
MTNR1B P49286 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
DRD2 P14416 4/20 0.32
DRD1 P21728 4/20 0.32
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
OPRM1 P35372 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11231949 0.82 ACHE (0.38) ACHENQO2MTNR1AMTNR1BMEN1
SCHEMBL11225535 0.82 ACHE (0.33) ACHENQO2MTNR1AMTNR1BMEN1
SCHEMBL11222326 0.82 NQO2 (0.33) ACHENQO2MTNR1AMTNR1BMEN1
SCHEMBL11224307 0.77 NQO2 (0.40) ACHENQO2MTNR1AMTNR1BMEN1
SCHEMBL11221371 0.76 ACHE (0.36) ACHENQO2MTNR1AMTNR1BMEN1
SCHEMBL11223892 0.72 PTGS2 (0.33) ACHEDRD2DRD1
SCHEMBL11223981 0.72 ACHE (0.37) ACHENQO2MTNR1AMTNR1BMEN1
SCHEMBL11225168 0.68 ATM (0.42) ACHEMEN1KMT2ADRD1NPC1
SCHEMBL11224305 0.68 NQO2 (0.37) ACHENQO2MTNR1AMTNR1BMEN1
SCHEMBL11219809 0.67 ACHE (0.35) ACHENQO2MTNR1AMTNR1BMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4352805-A BENZOXEPINE DERIVATIVES THE UPJOHN COMPANY (US) 1982-10-05 US disclosed
US-4312868-A HYPOTENSIVE, ANTIPSYCHOTIC THE UPJOHN COMPANY (US) 1982-01-26 US disclosed
US-4251526-A HYPOTENSIVE AGENTS AND ANTIPSYCHOTIC PHARMACIA & UPJOHN COMPANY 1981-02-17 US disclosed
US-4250181-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1981-02-10 US disclosed
US-4250175-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS PHARMACIA & UPJOHN COMPANY 1981-02-10 US disclosed
US-4247553-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1981-01-27 US disclosed
US-4179510-A ISOCHROMANS AND 2-BENZOXEPINS THE UPJOHN COMPANY (US) 1979-12-18 US disclosed
US-4166062-A HYPOTENSIVE AGENTS, CNS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1979-08-28 US disclosed
US-4153612-A 2-Benzoxepins THE UPJOHN COMPANY (US) 1979-05-08 US disclosed