SCHEMBL11224320

SCHEMBL11224320

CCOc1ccc2c(c1)CCCOC2COCCOS(=O)(=O)c1ccc(CC)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 5/20 0.39
CA9 Q16790 5/20 0.39
CA2 P00918 4/20 0.39
CA7 P43166 4/20 0.39
CA14 Q9ULX7 4/20 0.39
PPARA Q07869 4/20 0.38
PPARD Q03181 3/20 0.38
SMN1; SMN2 Q16637 3/20 0.35
ALDH1A1 P00352 2/20 0.35
HTT P42858 1/20 0.35
LMNA P02545 2/20 0.33
CA12 O43570 1/20 0.33
KDM4E B2RXH2 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
PPARG P37231 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11225262 0.81 CA1 (0.39) CA1CA9CA2CA7CA14
SCHEMBL11217850 0.80 PPARD (0.39) CA1CA9CA2CA7CA14
SCHEMBL11226510 0.80 PPARD (0.41) CA1CA9CA2CA7CA14
SCHEMBL11238280 0.75 ALDH1A1 (0.37) CA1CA9CA2CA7CA14
SCHEMBL11224385 0.73 PPARD (0.40) CA1CA9CA2CA7CA14
SCHEMBL11221009 0.72 PKM (0.37) CA1CA2SMN1; SMN2ALDH1A1HTT
SCHEMBL11218512 0.72 CA1 (0.44) CA1CA9CA2CA7CA14
SCHEMBL11218367 0.71 PPARD (0.39) CA1CA9CA2CA7CA14
SCHEMBL11219842 0.70 MEN1 (0.36) SMN1; SMN2MEN1MAPTKMT2A
SCHEMBL11223854 0.69 CA1 (0.38) CA1CA9CA2CA14ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4352805-A BENZOXEPINE DERIVATIVES THE UPJOHN COMPANY (US) 1982-10-05 US disclosed
US-4312868-A HYPOTENSIVE, ANTIPSYCHOTIC THE UPJOHN COMPANY (US) 1982-01-26 US disclosed
US-4251526-A HYPOTENSIVE AGENTS AND ANTIPSYCHOTIC PHARMACIA & UPJOHN COMPANY 1981-02-17 US disclosed
US-4250181-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1981-02-10 US disclosed
US-4250175-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS PHARMACIA & UPJOHN COMPANY 1981-02-10 US disclosed
US-4247553-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1981-01-27 US disclosed
US-4207239-A HYPOTENSIVE, ANTIPSYCHOTIC THE UPJOHN COMPANY (US) 1980-06-10 US disclosed
US-4206123-A INTERMEDIATES FOR HYPOTENSIVES MCCALL JOHN M (US) 1980-06-03 US disclosed
US-4181665-A INTERMEDIATES FOR AMINO DERIVATIVES POSSESSING HYPOTENSIVE AND CENTRAL NERVOUS SYSTEM ACTIVITY THE UPJOHN COMPANY (US) 1980-01-01 US disclosed
US-4179510-A ISOCHROMANS AND 2-BENZOXEPINS THE UPJOHN COMPANY (US) 1979-12-18 US disclosed
US-4166062-A HYPOTENSIVE AGENTS, CNS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1979-08-28 US disclosed
US-4153612-A 2-Benzoxepins THE UPJOHN COMPANY (US) 1979-05-08 US disclosed