SCHEMBL11224499

SCHEMBL11224499

COc1cc2c(cc1OC)C(c1ccc(F)cc1)(C(C)CCCl)OCC2

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.36
ABCB1 P08183 2/20 0.34
MAOB P27338 1/20 0.33
KCNH2 Q12809 3/20 0.33
TMEM97 Q5BJF2 3/20 0.33
SIGMAR1 Q99720 3/20 0.33
MAPK10 P53779 1/20 0.32
POLB P06746 1/20 0.32
GPBAR1 Q8TDU6 2/20 0.31
KDM4C Q9H3R0 1/20 0.31
MEN1 O00255 1/20 0.31
CXCR3 P49682 1/20 0.31
NFE2L2 Q16236 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11225377 0.95 KMT2A (0.35) KMT2AABCB1MAOBKCNH2TMEM97
SCHEMBL11223863 0.87 KMT2A (0.32) KMT2AABCB1MAOBKCNH2TMEM97
SCHEMBL11217805 0.84 KMT2A (0.34) KMT2AABCB1MAOBMAPK10KDM4C
SCHEMBL11224044 0.79 KMT2A (0.33) KMT2AABCB1MAOBMAPK10KDM4C
SCHEMBL11229451 0.77 ALDH1A1 (0.33) KMT2AKCNH2TMEM97SIGMAR1MEN1
SCHEMBL11536230 0.77 KMT2A (0.36) KMT2AABCB1MAOB
SCHEMBL11232418 0.77 KMT2A (0.36) KMT2AABCB1MAOBKCNH2TMEM97
SCHEMBL11224396 0.76 SLC6A4 (0.41) KCNH2SIGMAR1
SCHEMBL11223955 0.75 SLC6A4 (0.41) KCNH2SIGMAR1
SCHEMBL11230716 0.73 ALDH1A1 (0.34) KMT2AKCNH2TMEM97SIGMAR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4352805-A BENZOXEPINE DERIVATIVES THE UPJOHN COMPANY (US) 1982-10-05 US disclosed
US-4312868-A HYPOTENSIVE, ANTIPSYCHOTIC THE UPJOHN COMPANY (US) 1982-01-26 US disclosed
US-4251526-A HYPOTENSIVE AGENTS AND ANTIPSYCHOTIC PHARMACIA & UPJOHN COMPANY 1981-02-17 US disclosed
US-4250181-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1981-02-10 US disclosed
US-4250175-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS PHARMACIA & UPJOHN COMPANY 1981-02-10 US disclosed
US-4247553-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1981-01-27 US disclosed
US-4179510-A ISOCHROMANS AND 2-BENZOXEPINS THE UPJOHN COMPANY (US) 1979-12-18 US disclosed
US-4153612-A 2-Benzoxepins THE UPJOHN COMPANY (US) 1979-05-08 US disclosed