SCHEMBL11224612

SCHEMBL11224612

COc1cc([N+](=O)[O-])cc(C)c1C1C(=O)CCCC1=O

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.43
TDP1 Q9NUW8 3/20 0.39
ERN1 O75460 1/20 0.39
PKM P14618 1/20 0.37
ALDH1A1 P00352 7/20 0.36
KMT2A Q03164 3/20 0.36
LMNA P02545 3/20 0.36
CYP3A4 P08684 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
MAPT P10636 3/20 0.35
MEN1 O00255 1/20 0.35
TSHR P16473 1/20 0.35
GPR35 Q9HC97 1/20 0.35
CRHBP P24387 1/20 0.35
CRHR2 Q13324 1/20 0.35
NPSR1 Q6W5P4 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11231562 0.85 HTT (0.42) HTTTDP1ERN1PKMALDH1A1
SCHEMBL11217395 0.82 ALDH1A1 (0.47) HTTTDP1ALDH1A1KMT2ALMNA
SCHEMBL11220379 0.77 XDH (0.43) TDP1ALDH1A1KMT2ALMNACYP3A4
SCHEMBL17302850 0.74 USP2 (0.33) ALDH1A1KMT2ALMNAMEN1
SCHEMBL17302877 0.73 USP2 (0.32) ALDH1A1LMNA
SCHEMBL11220411 0.72 ALDH1A1 (0.50) TDP1ALDH1A1KMT2ASMN1; SMN2MAPT
SCHEMBL31405107 0.71 HTT (0.59) HTTTDP1ERN1PKMALDH1A1
SCHEMBL5159243 0.71 HTT (0.59) HTTTDP1ERN1PKMALDH1A1
SCHEMBL11215288 0.71 HTT (0.41) HTTTDP1ERN1PKMALDH1A1
SCHEMBL11422478 0.71 HTT (0.53) HTTTDP1ERN1PKMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0007243-B1 2-ARYL-1,3-CYCLOHEXANEDIONE COMPOUNDS AND ALKALI METAL SALTS, AMMONIUM SALTS AND ENOL ESTERS THEREOF, COMPOSITION AND METHOD OF CONTROLLING ACARINA ECTOPARASITES ON WARMBLOODED ANIMALS UNION CARBIDE CORPORATION (US) 1982-11-17 EP disclosed
US-4257858-A REACTING A CYCLOHEXA-1,3-DIONE-2-DIAZIDE WITH AN ARYL COMPOUND UNION CARBIDE CORPORATION (US) 1981-03-24 US disclosed
US-4256658-A CYCLIZATION, BASIC CATALYST UNION CARBIDE CORPORATION (US) 1981-03-17 US disclosed
US-4256657-A CYCLIZATION, ACID CATALYST UNION CARBIDE CORPORATION (US) 1981-03-17 US disclosed
US-4256659-A Method of preparing 2-aryl-1,3-cyclohexanedione compounds UNION CARBIDE CORPORATION (US) 1981-03-17 US disclosed
US-4209532-A Biocidal 2-aryl-1,3-cyclohexane dione compounds and alkali metal and ammonium salts thereof UNION CARBIDE CORPORATION (US) 1980-06-24 US disclosed
EP-0007243-A1 2-Aryl-1,3-cyclohexanedione compounds and alkali metal salts, ammonium salts and enol esters thereof, composition and method of controlling acarina ectoparasites on warmblooded animals UNION CARBIDE CORPORATION (US) 1980-01-23 EP disclosed
US-4175135-A Method of controlling acarina ectoparasites on warmblooded animals by orally administering to the animal an ectoparasitically effective amount of a 2-aryl-1,3-cyclohexanedione compound, and alkali metal salts, ammonium salts and enol esters thereof UNION CARBIDE CORPORATION (US) 1979-11-20 US disclosed