SCHEMBL11226037

SCHEMBL11226037

N/C(=C/S(=O)(=O)c1ccccc1)NCCSCc1ccon1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSMB5 P28074 1/20 0.38
ALDH1A1 P00352 13/20 0.37
POLB P06746 6/20 0.37
CYP2C9 P11712 3/20 0.37
CYP2C19 P33261 3/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2D6 P10635 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
RECQL P46063 1/20 0.37
LMNA P02545 3/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
HTT P42858 3/20 0.34
KMT2A Q03164 3/20 0.34
MEN1 O00255 2/20 0.34
NPC1 O15118 1/20 0.34
HPGD P15428 3/20 0.34
L3MBTL1 Q9Y468 2/20 0.33
BLM P54132 1/20 0.33
CYP1A2 P05177 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11226041 1.00 PSMB5 (0.38) PSMB5ALDH1A1POLBCYP2C9CYP2C19
SCHEMBL11225460 0.90 MAPT (0.38) ALDH1A1RECQLLMNASMN1; SMN2HTT
SCHEMBL11229742 0.90 ALDH1A1 (0.35) PSMB5ALDH1A1POLBCYP2C9CYP2C19
SCHEMBL11221306 0.86 PYGL (0.34) ALDH1A1POLBCYP2C9CYP2C19CYP3A4
SCHEMBL11232933 0.82 PSMB5 (0.38) PSMB5ALDH1A1POLBCYP2C9CYP2C19
SCHEMBL11232931 0.82 PSMB5 (0.38) PSMB5ALDH1A1POLBCYP2C9CYP2C19
SCHEMBL11633107 0.79 PSMB5 (0.34) PSMB5ALDH1A1POLBCYP2C9CYP2C19
SCHEMBL11633110 0.79 PSMB5 (0.34) PSMB5ALDH1A1POLBCYP2C9CYP2C19
SCHEMBL11231066 0.76 PSMB5 (0.39) PSMB5ALDH1A1POLBCYP2C9CYP2C19
SCHEMBL11667840 0.75 PSMB5 (0.67) PSMB5ALDH1A1POLBCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4317829-A ANTIHISTAMINES SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1982-03-02 US disclosed
US-4284640-A ANTIHISTAMINES SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1981-08-18 US disclosed
US-4277485-A INHIBITORS OF GASTRIC ACID SECRETION SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1981-07-07 US disclosed
US-4220652-A INHIBITORS OF H-2 HISTAMINE RECEPTORS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1980-09-02 US disclosed
US-4153704-A HETEROCYCLIC-ALKYL-AMINO SUBSTITUTED, ANTIHISTAMINES SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1979-05-08 US disclosed
US-4124717-A INHIBITORS OF H-2 HISTAMINE RECEPTORS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1978-11-07 US disclosed