SCHEMBL11226239

SCHEMBL11226239

C#Cc1cccc([N+](=O)[O-])c1.C1CC2CCC2C1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.46
TSHR P16473 3/20 0.46
ACHE P22303 2/20 0.42
ALDH1A1 P00352 5/20 0.42
MAPT P10636 2/20 0.42
HSP90AA1 P07900 2/20 0.42
S1PR2 O95136 1/20 0.42
OPRK1 P41145 1/20 0.42
HTT P42858 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
KDM1A O60341 1/20 0.41
POLB P06746 1/20 0.41
TDP1 Q9NUW8 1/20 0.40
ALOX15 P16050 1/20 0.40
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11237941 0.95 TSHR (0.50) LMNATSHRACHEALDH1A1MAPT
SCHEMBL11223757 0.90 TSHR (0.47) LMNATSHRACHEALDH1A1MAPT
SCHEMBL1477030 0.86 TSHR (0.61) LMNATSHRACHEALDH1A1MAPT
Methyl Alcohol SCHEMBL28555835 0.81 TSHR (0.55) LMNATSHRACHEALDH1A1MAPT
SCHEMBL11238907 0.79 VCAM1 (0.50) LMNATSHRALDH1A1HTTMEN1
SCHEMBL11239995 0.78 VCAM1 (0.37) TSHRALDH1A1TDP1MEN1KMT2A
SCHEMBL11443206 0.76 TSHR (0.53) LMNATSHRACHEALDH1A1MAPT
SCHEMBL11246750 0.73 MEN1 (0.38) TDP1MEN1KMT2A
SCHEMBL11240285 0.73 DRD2 (0.36) ALDH1A1KDM1AMEN1KMT2A
SCHEMBL11233082 0.73 DRD2 (0.43) TSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4150148-A NITROSUBSTITUTED WILLIAM H. RORER, INC. (US) 1979-04-17 US claimed
US-3981932-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1976-09-21 US claimed
US-4365093-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1982-12-21 US disclosed
US-4296264-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1981-10-20 US disclosed
US-4288457-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1981-09-08 US disclosed
US-4264627-A Ethynylbenzene compounds and derivatives thereof to treat inflammation, pain or fever WILLIAM H. RORER, INC. (US) 1981-04-28 US disclosed
US-4171373-A Ethynylbenzene compounds and derivatives thereof to treat pain, fever and inflammation WILLIAM H. RORER, INC. (US) 1979-10-16 US disclosed
US-4168320-A Ethynylbenzene compounds and derivatives thereof to treat inflammation, pain or fever WILLIAM H. RORER, INC. (US) 1979-09-18 US disclosed
US-4166133-A ETHYNYLBENZENE COMPOUNDS AND DERIVATIVES THEREOF TO TREAT PAIN, FEVER AND INFLAMMATION WILLIAM H. RORER, INC. (US) 1979-08-28 US disclosed
US-4157449-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1979-06-05 US disclosed
US-4150148-A NITROSUBSTITUTED WILLIAM H. RORER, INC. (US) 1979-04-17 US disclosed
US-4120889-A Cyano ethynylbenzene compounds WILLIAM H. RORER, INC. (US) 1978-10-17 US disclosed
US-4120885-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1978-10-17 US disclosed
US-4105786-A ANTIINFLAMMATORY WILLIAM H. RORER, INC. (US) 1978-08-08 US disclosed
US-4101591-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1978-07-18 US disclosed
US-4096279-A Ethynylbenzene compounds and derivatives thereof in the treatment of pain fever and inflammation WILLIAM H. RORER, INC. (US) 1978-06-20 US disclosed
US-4094995-A ETHYNYLBENZENE COMPOUNDS AND DERIVATIVES THEREOF TO TREAT PAIN, FEVER AND INFLAMMATION WILLIAM H. RORER, INC. (US) 1978-06-13 US disclosed
US-4093737-A Ethynylbenzene compounds and derivatives thereof in the treatment of pain, fever or inflammation WILLIAM H. RORER, INC. (US) 1978-06-06 US disclosed
US-4075354-A ETHYNYLBENZENE COMPOUNDS AND DERIVATIVES THEREOF FOR TREATING PAIN FEVER AND INFLAMMATION WILLIAM H. RORER, INC. (US) 1978-02-21 US disclosed
US-3981932-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1976-09-21 US disclosed