SCHEMBL11226436

SCHEMBL11226436

CC(CO)CNCCCOc1cccc2ccc(=O)[nH]c12

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 6/20 0.40
KDM4E B2RXH2 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
ADRB2 P07550 5/20 0.38
ADRB1 P08588 3/20 0.38
ALDH1A1 P00352 2/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HTR1B P28222 3/20 0.38
NR2E1 Q9Y466 1/20 0.38
MCHR1 Q99705 1/20 0.36
HTR1D P28221 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11858914 0.83 HTR1D (0.46) DRD2TDP1ALDH1A1KMT2AHTR1B
SCHEMBL11225424 0.82 HTR1B (0.43) DRD2KDM4ETDP1ADRB2ADRB1
Hydrochloric Acid SCHEMBL11230318 0.81 HTR1B (0.42) DRD2KDM4ETDP1ADRB2ADRB1
SCHEMBL11572052 0.81 DRD2 (0.57) DRD2KDM4ETDP1ADRB2ADRB1
SCHEMBL11864174 0.80 HTR1B (0.43) DRD2KDM4ETDP1ADRB2ADRB1
SCHEMBL11221461 0.79 ADRB2 (0.54) DRD2ADRB2ADRB1
SCHEMBL11872997 0.78 DRD2 (0.40) DRD2ADRB2ADRB1KMT2AHTR1B
SCHEMBL10064553 0.75 MCHR1 (0.48) DRD2TDP1HTR1BMCHR1
SCHEMBL11873001 0.75 KDM4E (0.38) DRD2KDM4EALDH1A1KMT2AHTR1B
SCHEMBL9820774 0.74 MCHR1 (0.49) TDP1KMT2AMEN1HTR1BMCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3953456-A ADRENERGIC BLOCKING AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JA) 1976-04-27 US claimed
US-4309432-A TOPICAL ADMINISTRATION OTSUKA PHARMACEUTICAL COMPANY, LTD. (JP) 1982-01-05 US disclosed
US-3953456-A ADRENERGIC BLOCKING AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JA) 1976-04-27 US disclosed