SCHEMBL11228515

SCHEMBL11228515

CN(C)c1nn(C)c2ncc(-c3cccnc3)cc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.52
CYP1A2 P05177 4/20 0.51
CYP3A4 P08684 4/20 0.51
CYP2C9 P11712 3/20 0.51
CYP2D6 P10635 3/20 0.51
CLK4 Q9HAZ1 3/20 0.51
LMNA P02545 2/20 0.51
MAPK1 P28482 2/20 0.51
HIF1A Q16665 1/20 0.51
FYN P06241 1/20 0.43
ALDH1A1 P00352 3/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
GLA P06280 1/20 0.41
TSHR P16473 1/20 0.41
CYP2A6 P11509 5/20 0.40
CYP2E1 P05181 1/20 0.40
CYP2B6 P20813 1/20 0.40
CYP2C19 P33261 1/20 0.40
CHEK1 O14757 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11232476 0.85 GSK3B (0.49) GSK3BCYP1A2CYP3A4MAPK1ALDH1A1
SCHEMBL11222259 0.82 GSK3B (0.76) GSK3BCYP1A2CYP3A4CYP2C9FYN
SCHEMBL11238844 0.73 GSK3B (0.45) GSK3BCYP1A2CYP3A4MAPK1ALDH1A1
SCHEMBL11233955 0.72 GSK3B (0.45) GSK3BCYP1A2CYP3A4CYP2C9CYP2D6
SCHEMBL19790564 0.72 GSK3B (0.36) GSK3BLMNAALOX15RXFP1
SCHEMBL11235819 0.72 CYP2C9 (0.38) GSK3BCYP1A2CYP3A4CYP2C9CYP2D6
SCHEMBL15081327 0.71 GSK3B (0.41) GSK3BCHEK1ALOX15
SCHEMBL11234318 0.71 GSK3B (0.46) GSK3BCYP1A2CYP3A4MAPK1ALDH1A1
SCHEMBL11233493 0.71 GSK3B (0.58) GSK3BCYP1A2MAPK1ALDH1A1MEN1
SCHEMBL22554308 0.69 GRM5 (0.47) GSK3BCYP2C9LMNACYP2A6CYP2E1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4361568-A 5-(Pyridinyl)-1H-pyrazolo[3,4-b]pyridin-3-amines and their cardiotonic use STERLING DRUG INC. (US) 1982-11-30 US disclosed
EP-0063754-A1 Pyrazolopyridine derivatives, and preparation, useful as cardiotonics STERLING DRUG INC. (US) 1982-11-03 EP disclosed