SCHEMBL11228623

SCHEMBL11228623

CCC(C)(C)NCC(O)COc1cccc(C)c1C

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.54
MAPT P10636 2/20 0.50
KDM4E B2RXH2 1/20 0.50
MEN1 O00255 1/20 0.50
ALDH1A1 P00352 1/20 0.50
KMT2A Q03164 1/20 0.50
ADRB2 P07550 4/20 0.49
ADRB1 P08588 3/20 0.49
ADRB3 P13945 2/20 0.49
GRK3 P35626 2/20 0.48
CASR P41180 2/20 0.48
NMT2 O60551 1/20 0.47
NMT1 P30419 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Xibenolol SCHEMBL79880 0.88 CYP2D6 (0.70) CYP2D6MAPTKDM4EMEN1ALDH1A1
Xibenolol SCHEMBL6506961 0.88 CYP2D6 (0.70) CYP2D6MAPTKDM4EMEN1ALDH1A1
Xibenolol SCHEMBL29387811 0.88 CYP2D6 (0.70) CYP2D6MAPTKDM4EMEN1ALDH1A1
Xibenolol SCHEMBL79879 0.88 CYP2D6 (0.70) CYP2D6MAPTKDM4EMEN1ALDH1A1
Xibenolol SCHEMBL7267198 0.86 CYP2D6 (0.72) CYP2D6MAPTKDM4EMEN1ALDH1A1
SCHEMBL11855803 0.81 CASR (0.70) CYP2D6MAPTKDM4EADRB2ADRB1
SCHEMBL3956865 0.80 ALOX15 (0.63) CYP2D6KDM4EMEN1ALDH1A1KMT2A
SCHEMBL11223419 0.78 ADRB2 (0.62) CYP2D6MAPTKDM4EMEN1KMT2A
SCHEMBL10893056 0.78 GRK3 (0.49) CYP2D6MAPTKDM4EMEN1ALDH1A1
Hydrochloric Acid SCHEMBL9506677 0.78 KMT2A (0.50) CYP2D6KDM4EMEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4360464-A Process for production of 1-aryloxy-aminopropane derivatives TEIKOKU HORMONE MFG. CO. LTD. (JP) 1982-11-23 US disclosed
US-4018824-A ANTIULCER AND ADRENERGIC BLOCKING AGENTS TEIKOKU HORMONE MFG. CO., LTD. (JA) 1977-04-19 US disclosed