SCHEMBL11229010

SCHEMBL11229010

CCOC(=O)C1CCc2c(sc3ccc(C)cc23)C1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LIMK1 P53667 1/20 0.53
MAPT P10636 3/20 0.50
POLB P06746 2/20 0.50
PDK1 Q15118 1/20 0.46
MKNK1 Q9BUB5 1/20 0.42
P2RX3 P56373 1/20 0.42
KDM4E B2RXH2 2/20 0.39
TP53 P04637 1/20 0.38
LGMN Q99538 1/20 0.38
ALDH1A1 P00352 3/20 0.38
HPGD P15428 2/20 0.38
MDM2 Q00987 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
TSHR P16473 2/20 0.37
GAA P10253 1/20 0.37
ALOX15 P16050 1/20 0.37
ALOX12 P18054 1/20 0.37
HSD17B10 Q99714 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11789706 0.89 LIMK1 (0.57) LIMK1MAPTPOLBPDK1MKNK1
SCHEMBL11795888 0.89 LIMK1 (0.52) LIMK1MAPTPOLBPDK1MKNK1
SCHEMBL11246538 0.86 LIMK1 (0.55) LIMK1MAPTPDK1MKNK1P2RX3
SCHEMBL11786639 0.84 MAPT (0.38) LIMK1MAPTPOLBPDK1P2RX3
SCHEMBL4905684 0.82 LIMK1 (0.52) LIMK1MAPTPOLBPDK1MKNK1
SCHEMBL4904247 0.80 ALDH1A1 (0.43) LIMK1MAPTPOLBPDK1MKNK1
SCHEMBL4905260 0.80 PDK1 (0.42) LIMK1MAPTPOLBPDK1MKNK1
SCHEMBL11810317 0.78 LIMK1 (0.44) LIMK1MAPTPOLBPDK1MKNK1
SCHEMBL4895798 0.77 ALDH1A1 (0.40) LIMK1MAPTPOLBPDK1MKNK1
SCHEMBL4904164 0.76 PDK1 (0.46) LIMK1MAPTPDK1KDM4ETP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4334078-A ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTIRHEUMATICS HOFFMANN-LA ROCHE INC. (US) 1982-06-08 US disclosed
US-4219657-A USED AS ANTIINFLAMATORY AGENTS, ANALGESICS, ANTIRHEUMATIC AGENTS HOFFMANN-LA ROCHE INC. (US) 1980-08-26 US disclosed