SCHEMBL11229680

SCHEMBL11229680

COc1ccc(C2CN(CC3CC3)CCc3c2cc(OC)c(OC)c3Cl)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 6/20 0.39
DRD2 P14416 5/20 0.39
DRD4 P21917 1/20 0.39
DRD5 P21918 1/20 0.39
DRD3 P35462 1/20 0.39
KDM2B Q8NHM5 2/20 0.39
MTOR P42345 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
ALOX15 P16050 1/20 0.37
NFKB1 P19838 1/20 0.37
THPO P40225 1/20 0.37
HIF1A Q16665 1/20 0.37
HSD17B10 Q99714 1/20 0.37
KDM4E B2RXH2 1/20 0.37
GMNN O75496 1/20 0.37
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11216105 0.85 DRD1 (0.50) DRD1DRD2DRD5MTORCYP1A2
SCHEMBL11283177 0.85 DRD2 (0.56) DRD1DRD2DRD4DRD5DRD3
SCHEMBL11309660 0.83 HRH3 (0.37) DRD1DRD2KDM2BMTORCYP1A2
Hydrochloric Acid SCHEMBL11253560 0.83 KDM2B (0.38) DRD2KDM2B
Bromide SCHEMBL11242453 0.83 KDM2B (0.37) KDM2BCYP3A4CYP2D6
Bromide SCHEMBL11236726 0.79 DRD2 (0.38) DRD1DRD2DRD4DRD5DRD3
Hydrochloric Acid SCHEMBL11262602 0.78 BCHE (0.50) DRD1DRD2MTORCYP1A2CYP3A4
SCHEMBL13928827 0.77 DRD1 (0.50) DRD1DRD2DRD5MTORCYP1A2
SCHEMBL11529724 0.76 DRD1 (0.46) DRD1DRD2MTORCYP1A2CYP3A4
SCHEMBL7322313 0.76 CYP2D6 (0.63) DRD1DRD2DRD5MTORCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4328153-A HYPOTENSIVE AGENT SMITH KLINE CORPORATION (US) 1982-05-04 US disclosed
EP-0044709-A1 New dopaminergic benzazepines SMITHKLINE BECKMAN CORPORATION (US) 1982-01-27 EP disclosed