SCHEMBL11230718

SCHEMBL11230718

COc1cc2c(cc1OC)C(C)(CCC(C)Cl)OCCC2

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 2/20 0.34
KDM4E B2RXH2 3/20 0.32
ALDH1A1 P00352 2/20 0.32
MAPK1 P28482 2/20 0.32
GLA P06280 1/20 0.32
HPGD P15428 1/20 0.32
KCNH2 Q12809 2/20 0.32
TMEM97 Q5BJF2 2/20 0.32
SIGMAR1 Q99720 2/20 0.32
ALOX5 P09917 1/20 0.30
MEN1 O00255 1/20 0.30
MAPT P10636 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11225472 0.82 MAPK1 (0.33) AKT1KDM4EALDH1A1MAPK1MEN1
SCHEMBL11220983 0.81 MAPK1 (0.33) AKT1KDM4EALDH1A1MAPK1MEN1
SCHEMBL11230716 0.76 ALDH1A1 (0.34) AKT1KDM4EALDH1A1MAPK1GLA
SCHEMBL11219802 0.74 MAPT (0.33) AKT1KDM4EALDH1A1MAPK1MEN1
SCHEMBL11220851 0.73 MAPT (0.32) AKT1KDM4EALDH1A1MAPK1MEN1
SCHEMBL11223876 0.73 ALDH1A1 (0.32) ALDH1A1MAPK1
SCHEMBL11536230 0.73 KMT2A (0.36) KMT2A
SCHEMBL11221731 0.71 ALOX15 (0.39) KDM4EALDH1A1MAPK1MEN1MAPT
SCHEMBL11226312 0.70 ALDH1A1 (0.32) AKT1ALDH1A1MAPK1MAPT
SCHEMBL11265594 0.70 HSD17B10 (0.40) KDM4EALDH1A1MAPK1MEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4352805-A BENZOXEPINE DERIVATIVES THE UPJOHN COMPANY (US) 1982-10-05 US disclosed
US-4312868-A HYPOTENSIVE, ANTIPSYCHOTIC THE UPJOHN COMPANY (US) 1982-01-26 US disclosed
US-4251526-A HYPOTENSIVE AGENTS AND ANTIPSYCHOTIC PHARMACIA & UPJOHN COMPANY 1981-02-17 US disclosed
US-4250181-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1981-02-10 US disclosed
US-4250175-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS PHARMACIA & UPJOHN COMPANY 1981-02-10 US disclosed
US-4247553-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1981-01-27 US disclosed
US-4179510-A ISOCHROMANS AND 2-BENZOXEPINS THE UPJOHN COMPANY (US) 1979-12-18 US disclosed
US-4153612-A 2-Benzoxepins THE UPJOHN COMPANY (US) 1979-05-08 US disclosed