SCHEMBL11235747

SCHEMBL11235747

CCCCCc1[nH]c(=O)c(Cl)cc1-c1ccncc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 5/20 0.55
PDE3A Q14432 5/20 0.55
GSK3B P49841 2/20 0.43
GPR84 Q9NQS5 5/20 0.39
AURKB Q96GD4 1/20 0.39
INCENP Q9NQS7 1/20 0.39
APLNR P35414 1/20 0.37
KDM4E B2RXH2 1/20 0.36
PDE5A O76074 1/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
PTGS1 P23219 1/20 0.36
PDE4A P27815 1/20 0.36
CYP2C19 P33261 1/20 0.36
BLM P54132 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
CDK5 Q00535 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11245033 0.91 PDE3B (0.66) PDE3BPDE3AGSK3BAURKBINCENP
SCHEMBL11238746 0.85 PDE3B (0.64) PDE3BPDE3AGSK3BAURKBINCENP
SCHEMBL11229942 0.84 PDE3B (0.58) PDE3BPDE3AGSK3BGPR84AURKB
SCHEMBL11118932 0.81 PDE3B (0.57) PDE3BPDE3AGSK3BAURKBINCENP
SCHEMBL11224748 0.81 PDE3A (0.84) PDE3BPDE3AGSK3BGPR84AURKB
SCHEMBL11247774 0.81 PDE3B (0.52) PDE3BPDE3AGSK3BGPR84APLNR
SCHEMBL11242743 0.81 PDE3B (0.54) PDE3BPDE3AGSK3BGPR84AURKB
SCHEMBL11249495 0.80 PDE3B (0.51) PDE3BPDE3AGSK3BGPR84AURKB
SCHEMBL11235237 0.80 PDE3B (0.51) PDE3BPDE3AGSK3BGPR84AURKB
SCHEMBL11236384 0.80 PDE3B (0.56) PDE3BPDE3AGSK3BGPR84AURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4365065-A 1-(Pyridinyl)-2-(dimethylamino)ethenyl lower-alkyl ketones STERLING DRUG INC. (US) 1982-12-21 US disclosed
US-4313951-A 3-Substituted-6-(lower-alkyl)-5-(pyridinyl)-2(1H)-pyridinones, their cardiotonic use and intermediates therefor STERLING DRUG INC. (US) 1982-02-02 US disclosed